SCHEMBL8306394

SCHEMBL8306394

NC(=O)/C=C(\N[C@H](C(N)=O)c1ccccc1)c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 1/20 0.40
CYP3A4 P08684 3/20 0.40
TSHR P16473 2/20 0.40
ALDH1A1 P00352 1/20 0.40
CYP1A2 P05177 1/20 0.40
ROCK2 O75116 3/20 0.39
ROCK1 Q13464 2/20 0.39
CNR1 P21554 1/20 0.38
GPR88 Q9GZN0 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CYP2C9 P11712 1/20 0.37
PDGFRA P16234 1/20 0.37
MAPK1 P28482 1/20 0.37
MAPKAPK2 P49137 1/20 0.37
RPS6KA1 Q15418 1/20 0.37
AURKB Q96GD4 1/20 0.37
CSNK1G1 Q9HCP0 1/20 0.37
LMNA P02545 4/20 0.37
HPGD P15428 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8302401 0.85 GPR88 (0.40) TACR3CYP3A4TSHRALDH1A1CYP1A2
SCHEMBL8303024 0.80 LTB4R (0.48) TSHRALDH1A1CYP1A2CYP2C9MAPK1
SCHEMBL8303022 0.78 ALDH1A1 (0.46) CYP3A4ALDH1A1CA1CA2TDP1
SCHEMBL10332571 0.76 LMNA (0.53) TACR3CYP3A4ALDH1A1ROCK2ROCK1
SCHEMBL22502277 0.76 LMNA (0.49) TACR3CYP3A4ROCK2ROCK1CNR1
SCHEMBL4732145 0.76 LMNA (0.49) TACR3CYP3A4ROCK2ROCK1CNR1
SCHEMBL8303023 0.75 CNR2 (0.49) ALDH1A1CNR1HPGDMAPTEPHX1
SCHEMBL8302370 0.75 CYP3A4 (0.48) CYP3A4TSHRALDH1A1CYP1A2CNR1
SCHEMBL12880512 0.73 LMNA (0.46) TACR3CYP3A4ROCK2ROCK1CNR1
SCHEMBL13707805 0.73 TACR3 (0.46) TACR3CYP3A4ROCK2ROCK1CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004085661-A2 PROCESS TO CHIRAL BETA-AMINO ACID DERIVATIVES MERCK & CO., INC (US) 2004-10-07 WO disclosed