SCHEMBL8303024

SCHEMBL8303024

NC(=O)[C@@H](N/C(=C\C(=O)N1CCCCC1)c1ccccc1)c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTB4R Q15722 1/20 0.48
LTB4R2 Q9NPC1 1/20 0.48
HPGD P15428 4/20 0.42
GAA P10253 2/20 0.41
KMT2A Q03164 5/20 0.39
MAPT P10636 2/20 0.39
KDM4E B2RXH2 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
GFER P55789 1/20 0.39
ALDH1A1 P00352 2/20 0.39
USP2 O75604 1/20 0.39
F10 P00742 4/20 0.39
PRSS1 P07477 4/20 0.39
F2 P00734 3/20 0.39
MEN1 O00255 2/20 0.39
CYP2C9 P11712 2/20 0.39
PARP1 P09874 1/20 0.38
PARP15 Q460N3 1/20 0.38
PARP10 Q53GL7 1/20 0.38
TSHR P16473 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8306394 0.80 TACR3 (0.40) HPGDMAPTALDH1A1CYP2C9PARP1
SCHEMBL8305615 0.80 CNR2 (0.46) LTB4RLTB4R2HPGDGAAKMT2A
SCHEMBL8302401 0.76 GPR88 (0.40) GAAKMT2AMAPTKDM4EALDH1A1
SCHEMBL8303022 0.69 ALDH1A1 (0.46) GAAKMT2AMAPTKDM4EALDH1A1
SCHEMBL8306001 0.68 HPGD (0.49) HPGDGAAKMT2AALDH1A1MEN1
SCHEMBL4732145 0.67 LMNA (0.49) GAACYP2C9MAPK1
SCHEMBL22502277 0.67 LMNA (0.49) GAACYP2C9MAPK1
SCHEMBL10332571 0.67 LMNA (0.53) GAAALDH1A1CYP2C9MAPK1
SCHEMBL16339449 0.66 KLRK1 (0.48) HPGDGAAKMT2AMAPTKDM4E
SCHEMBL23716017 0.65 LMNA (0.65) HPGDKMT2AALDH1A1MEN1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004085661-A2 PROCESS TO CHIRAL BETA-AMINO ACID DERIVATIVES MERCK & CO., INC (US) 2004-10-07 WO disclosed