SCHEMBL8315899

SCHEMBL8315899

O=C(Cl)Oc1ccc(I)cc1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TPMT P51580 1/20 0.41
CA1 P00915 4/20 0.40
CA2 P00918 4/20 0.40
CA9 Q16790 2/20 0.40
RXRA P19793 1/20 0.39
RXRB P28702 1/20 0.39
RAB9A P51151 1/20 0.38
HRH3 Q9Y5N1 1/20 0.37
CA12 O43570 1/20 0.37
APP P05067 4/20 0.37
LMNA P02545 1/20 0.37
GSK3B P49841 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6924446 0.87 RAB9A (0.46) RAB9ALMNA
SCHEMBL6564201 0.80 ELANE (0.52) RAB9ALMNA
SCHEMBL6565732 0.80 HSD17B10 (0.47) RAB9ALMNA
SCHEMBL7866352 0.80 MEN1 (0.50) TPMTCA1CA2CA9RXRA
SCHEMBL59462 0.78 ELANE (0.48)
SCHEMBL9578961 0.78 MAPT (0.50) CA1CA2CA9RAB9ACA12
SCHEMBL7871721 0.78 TPMT (0.48) TPMTCA1CA2CA9RXRA
SCHEMBL1268683 0.76 LDHA (0.47) CA1CA2CA9RXRARXRB
SCHEMBL3292329 0.76 ALDH1A1 (0.43) RAB9A
SCHEMBL696908 0.76 KMT2A (0.44) CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10870706-B2 Bifunctional cytotoxic agents containing the CTI pharmacophore PFIZER INC. (US) 2020-12-22 US disclosed
US-9598410-B2 Substituted 4,5,6,7-tetrahydro-1H-pyrazolo[4,3-C]pyridines, their use as medicament, and pharmaceutical preparations comprising them SANOFI (FR) 2017-03-21 US disclosed
WO-2004058754-A1 BENZOAZOLYPIPERAZINE DERIVATIVES HAVING MGLUR1- AND MGLUR5-ANTAGONISTIC ACTIVITY EURO-CELTIQUE S.A. (LU) 2004-07-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10870706-B2 Bifunctional cytotoxic agents containing the CTI pharmacophore CCNI, TTI1, TTI2 TPMT 3188/4885CA1 1228/4885CA2 1071/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.