SCHEMBL8323592

SCHEMBL8323592

CN(C)C([CH]c1ccc(F)cc1)Cc1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.40
NOS1 P29475 1/20 0.40
NOS2 P35228 1/20 0.40
NFE2L2 Q16236 1/20 0.40
PPARG P37231 1/20 0.38
PPARA Q07869 1/20 0.38
ADRA2B P18089 1/20 0.38
ADRA2C P18825 1/20 0.38
SLC6A2 P23975 1/20 0.38
HTR2A P28223 1/20 0.38
SLC6A4 P31645 1/20 0.38
ADRA1A P35348 1/20 0.38
OPRK1 P41145 1/20 0.38
SLC6A3 Q01959 1/20 0.38
KCNH2 Q12809 1/20 0.38
ALDH1A1 P00352 3/20 0.37
MAPT P10636 2/20 0.37
ALOX15 P16050 1/20 0.37
TSHR P16473 1/20 0.37
RECQL P46063 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8325718 0.85 CYP2C19 (0.40) PPARGPPARAADRA2BADRA2CSLC6A2
SCHEMBL8322987 0.83 NPC1 (0.52) NOS3NOS1NOS2PPARGPPARA
SCHEMBL8324481 0.83 NFE2L2 (0.45) NFE2L2PPARGPPARASLC6A2SLC6A4
SCHEMBL8324438 0.81 G6PC1 (0.48) PPARGPPARASLC6A4ALDH1A1MAPT
SCHEMBL8323270 0.80 KDM4E (0.36) NOS2PPARGPPARAADRA2BADRA2C
SCHEMBL8326594 0.78 NFE2L2 (0.44) NOS3NOS1NOS2NFE2L2PPARG
SCHEMBL8324682 0.75 TP53 (0.40) PPARGPPARAADRA2BADRA2CSLC6A2
SCHEMBL8324972 0.74 TAAR1 (0.44) NOS3NOS1NOS2NFE2L2PPARG
SCHEMBL8326976 0.74 MAOB (0.45) ADRA2BADRA2CSLC6A2HTR2ASLC6A4
SCHEMBL8327755 0.74 PNMT (0.41) ALDH1A1TSHRRECQLGRIN1GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0948496-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDONE COMPOUNDS AND METHODS OF USE Amgen inc. (US) 1999-10-13 EP disclosed
WO-1998024780-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDINONE COMPOUNDS AND THEIR USE AMGEN INC. (US) 1998-06-11 WO disclosed