SCHEMBL8324972

SCHEMBL8324972

CNC([CH]c1ccc(F)cc1)Cc1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 3/20 0.44
SLC18A2 Q05940 1/20 0.44
SIGMAR1 Q99720 1/20 0.44
NOS3 P29474 1/20 0.43
NOS1 P29475 1/20 0.43
NOS2 P35228 1/20 0.43
NFE2L2 Q16236 1/20 0.40
ALDH1A1 P00352 5/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
GRIN1 Q05586 1/20 0.39
GRIN2B Q13224 1/20 0.39
PPARG P37231 1/20 0.38
PPARA Q07869 1/20 0.38
POLB P06746 1/20 0.37
MAPT P10636 2/20 0.37
ALOX15 P16050 1/20 0.37
TSHR P16473 1/20 0.37
RECQL P46063 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8325444 0.85 TAAR1 (0.46) TAAR1SLC18A2SIGMAR1SMN1; SMN2PPARG
SCHEMBL8326774 0.83 NPC1 (0.52) TAAR1SLC18A2SIGMAR1NOS3NOS1
SCHEMBL8322850 0.83 NFE2L2 (0.45) TAAR1SLC18A2SIGMAR1NFE2L2PPARG
SCHEMBL8323399 0.81 LTA4H (0.50) TAAR1SLC18A2SIGMAR1ALDH1A1PPARG
SCHEMBL8322029 0.80 CYP3A4 (0.40) TAAR1SLC18A2SIGMAR1NOS2SMN1; SMN2
SCHEMBL8326594 0.78 NFE2L2 (0.44) TAAR1SLC18A2SIGMAR1NOS3NOS1
SCHEMBL8327429 0.75 TAAR1 (0.42) TAAR1SLC18A2SIGMAR1ALDH1A1POLB
SCHEMBL8323592 0.74 NOS3 (0.40) SIGMAR1NOS3NOS1NOS2NFE2L2
SCHEMBL8324981 0.74 GRIN1 (0.43) TAAR1SLC18A2SIGMAR1ALDH1A1GRIN1
SCHEMBL8325015 0.74 MAOA (0.45) TAAR1SLC18A2SIGMAR1MAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0948496-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDONE COMPOUNDS AND METHODS OF USE Amgen inc. (US) 1999-10-13 EP disclosed
WO-1998024780-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDINONE COMPOUNDS AND THEIR USE AMGEN INC. (US) 1998-06-11 WO disclosed