SCHEMBL8322987

SCHEMBL8322987

CN(C)C([CH]c1ccc(C(F)(F)F)cc1)Cc1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.52
RAB9A P51151 1/20 0.52
NOS3 P29474 1/20 0.44
NOS1 P29475 1/20 0.44
NOS2 P35228 1/20 0.44
PPARG P37231 1/20 0.42
PPARA Q07869 1/20 0.42
MTOR P42345 1/20 0.40
SLC6A9 P48067 1/20 0.39
MAPT P10636 2/20 0.39
FPR2 P25090 1/20 0.39
LMNA P02545 1/20 0.39
MAPK1 P28482 1/20 0.39
OPRM1 P35372 1/20 0.38
OPRL1 P41146 1/20 0.38
SLC6A4 P31645 1/20 0.37
HRH3 Q9Y5N1 1/20 0.37
ALDH1A1 P00352 1/20 0.37
TSHR P16473 1/20 0.37
BCHE P06276 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8322396 0.85 HTR2A (0.46) NPC1RAB9APPARGPPARAMAPT
SCHEMBL8323592 0.83 NOS3 (0.40) NOS3NOS1NOS2PPARGPPARA
SCHEMBL8325718 0.81 CYP2C19 (0.40) PPARGPPARAMAPTLMNASLC6A4
SCHEMBL8326251 0.80 NPC1 (0.59) NPC1RAB9ANOS3NOS1NOS2
SCHEMBL8324438 0.78 G6PC1 (0.48) PPARGPPARAMAPTOPRM1SLC6A4
SCHEMBL8326774 0.77 NPC1 (0.52) NPC1RAB9ANOS3NOS1NOS2
SCHEMBL8324481 0.73 NFE2L2 (0.45) NPC1RAB9APPARGPPARAMAPK1
SCHEMBL8323270 0.73 KDM4E (0.36) NOS2PPARGPPARAMAPTSLC6A4
SCHEMBL8324682 0.72 TP53 (0.40) NPC1PPARGPPARASLC6A4ALDH1A1
SCHEMBL8326976 0.71 MAOB (0.45) NPC1MAPTSLC6A4SIGMAR1HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0948496-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDONE COMPOUNDS AND METHODS OF USE Amgen inc. (US) 1999-10-13 EP disclosed
WO-1998024780-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDINONE COMPOUNDS AND THEIR USE AMGEN INC. (US) 1998-06-11 WO disclosed