SCHEMBL8324318

SCHEMBL8324318

Cc1cccc([CH]C(C)Cc2ccccc2)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 4/20 0.44
SLC6A2 P23975 2/20 0.44
SIGMAR1 Q99720 2/20 0.44
MAOA P21397 1/20 0.44
SLC6A4 P31645 1/20 0.44
SLC6A3 Q01959 1/20 0.44
CYP2A6 P11509 1/20 0.44
ADORA2A P29274 1/20 0.44
ADORA1 P30542 1/20 0.44
TP53 P04637 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
NPC1 O15118 1/20 0.42
CASP3 P42574 1/20 0.42
SENP8 Q96LD8 1/20 0.42
SENP7 Q9BQF6 1/20 0.42
SENP6 Q9GZR1 1/20 0.42
BACE1 P56817 1/20 0.40
ACHE P22303 1/20 0.39
BCHE P06276 1/20 0.39
PPARG P37231 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8323856 0.82 MAOA (0.49) TAAR1SLC6A2SIGMAR1MAOASLC6A4
SCHEMBL8324358 0.82 TAAR1 (0.43) TAAR1SLC6A2SIGMAR1MAOASLC6A4
SCHEMBL8319052 0.82 PNMT (0.49) TAAR1SLC6A2SIGMAR1MAOASLC6A4
SCHEMBL8330718 0.82 NFE2L2 (0.49) TAAR1SLC6A2SIGMAR1MAOASLC6A4
SCHEMBL8327667 0.81 TAAR1 (0.44) TAAR1SLC6A2SIGMAR1MAOASLC6A4
SCHEMBL8324682 0.80 TP53 (0.40) TAAR1SLC6A2SIGMAR1MAOASLC6A4
SCHEMBL8327429 0.80 TAAR1 (0.42) TAAR1SLC6A2SIGMAR1MAOASLC6A4
SCHEMBL8320387 0.78 HTR2A (0.53) TAAR1SLC6A2SIGMAR1SLC6A4SLC6A3
SCHEMBL18378693 0.74 TP53 (0.56) MAOATP53TDP1NPC1CASP3
SCHEMBL9346803 0.72 SLC6A2 (0.46) TAAR1SLC6A2SIGMAR1MAOASLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0948496-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDONE COMPOUNDS AND METHODS OF USE Amgen inc. (US) 1999-10-13 EP disclosed
WO-1998024780-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDINONE COMPOUNDS AND THEIR USE AMGEN INC. (US) 1998-06-11 WO disclosed