SCHEMBL8327667

SCHEMBL8327667

Cc1ccc([CH]C(C)Cc2ccccc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 5/20 0.44
SIGMAR1 Q99720 4/20 0.44
SLC6A2 P23975 2/20 0.44
MAOA P21397 1/20 0.44
SLC6A4 P31645 1/20 0.44
SLC6A3 Q01959 1/20 0.44
CYP2A6 P11509 1/20 0.44
ADORA2A P29274 1/20 0.44
ADORA1 P30542 1/20 0.44
SLC18A2 Q05940 1/20 0.41
CYP2D6 P10635 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
PLA2G1B P04054 1/20 0.40
POLB P06746 1/20 0.40
MAPT P10636 1/20 0.40
ATG4B Q9Y4P1 1/20 0.40
TRPA1 O75762 1/20 0.40
HTT P42858 1/20 0.39
CYP2C19 P33261 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8326594 0.84 NFE2L2 (0.44) TAAR1SIGMAR1SLC6A2MAOASLC6A4
SCHEMBL8324318 0.81 TAAR1 (0.44) TAAR1SIGMAR1SLC6A2MAOASLC6A4
SCHEMBL8323072 0.81 TRPA1 (0.50) SIGMAR1SLC6A4MEN1KMT2AMAPT
SCHEMBL8326251 0.80 NPC1 (0.59) TAAR1SIGMAR1SLC6A2MAOASLC6A4
SCHEMBL8325444 0.77 TAAR1 (0.46) TAAR1SIGMAR1SLC6A2MAOASLC6A4
SCHEMBL8325718 0.77 CYP2C19 (0.40) TAAR1SIGMAR1SLC6A2MAOASLC6A4
SCHEMBL9346803 0.76 SLC6A2 (0.46) TAAR1SIGMAR1SLC6A2MAOASLC6A4
SCHEMBL8327003 0.73 TRPA1 (0.38) TAAR1SIGMAR1SLC6A2MAOASLC6A4
SCHEMBL8323856 0.73 MAOA (0.49) TAAR1SIGMAR1SLC6A2MAOASLC6A4
SCHEMBL8319052 0.73 PNMT (0.49) TAAR1SIGMAR1SLC6A2MAOASLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0948496-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDONE COMPOUNDS AND METHODS OF USE Amgen inc. (US) 1999-10-13 EP disclosed
WO-1998024780-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDINONE COMPOUNDS AND THEIR USE AMGEN INC. (US) 1998-06-11 WO disclosed