SCHEMBL8319052

SCHEMBL8319052

CC([CH]c1cccc(Cl)c1)Cc1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PNMT P11086 1/20 0.49
SLC6A2 P23975 2/20 0.43
TAAR1 Q96RJ0 2/20 0.43
SIGMAR1 Q99720 2/20 0.43
MAOA P21397 1/20 0.43
SLC6A4 P31645 1/20 0.43
SLC6A3 Q01959 1/20 0.43
CYP2A6 P11509 1/20 0.43
ADORA2A P29274 1/20 0.43
ADORA1 P30542 1/20 0.43
GRIN1 Q05586 2/20 0.43
GRIN2B Q13224 2/20 0.43
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
ALDH1A1 P00352 2/20 0.41
HPGD P15428 1/20 0.41
CHRM5 P08912 1/20 0.41
SCN4A P35499 1/20 0.40
MEN1 O00255 1/20 0.39
LMNA P02545 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8324318 0.82 TAAR1 (0.44) SLC6A2TAAR1SIGMAR1MAOASLC6A4
SCHEMBL8324358 0.81 TAAR1 (0.43) SLC6A2TAAR1SIGMAR1MAOASLC6A4
SCHEMBL8323856 0.81 MAOA (0.49) SLC6A2TAAR1SIGMAR1MAOASLC6A4
SCHEMBL8330718 0.81 NFE2L2 (0.49) SLC6A2TAAR1SIGMAR1MAOASLC6A4
SCHEMBL8327755 0.80 PNMT (0.41) PNMTTAAR1SIGMAR1GRIN1GRIN2B
SCHEMBL8324981 0.80 GRIN1 (0.43) PNMTTAAR1SIGMAR1GRIN1GRIN2B
SCHEMBL8327003 0.80 TRPA1 (0.38) PNMTSLC6A2TAAR1SIGMAR1MAOA
SCHEMBL8320387 0.77 HTR2A (0.53) SLC6A2TAAR1SIGMAR1SLC6A4SLC6A3
SCHEMBL18243444 0.75 CHRM5 (0.52) PNMTGRIN1GRIN2BALDH1A1CHRM5
SCHEMBL3335734 0.73 CHRM5 (0.50) PNMTGRIN1GRIN2BCHRM5MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0948496-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDONE COMPOUNDS AND METHODS OF USE Amgen inc. (US) 1999-10-13 EP disclosed
WO-1998024780-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDINONE COMPOUNDS AND THEIR USE AMGEN INC. (US) 1998-06-11 WO disclosed