SCHEMBL8323939

SCHEMBL8323939

O=[N+]([O-])c1ccc(N(Cc2ccc(F)cc2)c2cncnc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 4/20 0.49
ESR1 P03372 1/20 0.47
ESR2 Q92731 1/20 0.47
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
KCNJ1 P48048 1/20 0.43
KCNH2 Q12809 1/20 0.43
CRHBP P24387 1/20 0.42
CRHR2 Q13324 1/20 0.42
MMP1 P03956 2/20 0.41
MMP2 P08253 2/20 0.41
MMP9 P14780 2/20 0.41
MMP8 P22894 2/20 0.41
MMP13 P45452 2/20 0.41
HSPB1 P04792 1/20 0.41
CYP19A1 P11511 1/20 0.41
NR1D1 P20393 1/20 0.41
NR1H3 Q13133 1/20 0.41
POLB P06746 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8327952 0.93 CRHBP (0.47) ARCRHBPCRHR2CYP19A1POLB
SCHEMBL8327623 0.87 ALDH1A1 (0.50) ARNPC1RAB9ACRHBPCRHR2
SCHEMBL8327171 0.87 CRHBP (0.42) ARCRHBPCRHR2CYP19A1POLB
SCHEMBL8326188 0.87 CYP19A1 (0.55) ARNPC1RAB9ACRHBPCRHR2
SCHEMBL8329070 0.86 MMP1 (0.45) ARRAB9ACRHBPCRHR2MMP1
SCHEMBL8324619 0.84 KCNJ1 (0.46) ARNPC1KCNJ1KCNH2CRHBP
SCHEMBL8323517 0.84 KCNJ1 (0.46) ARNPC1KCNJ1KCNH2CRHBP
SCHEMBL3737073 0.77 KCNJ1 (0.51) ARNPC1RAB9AKCNJ1KCNH2
SCHEMBL8323103 0.76 ESR1 (0.49) ESR1ESR2CYP19A1NR1D1MAOB
SCHEMBL8327951 0.72 SLC29A1 (0.41) NPC1RAB9AHSPB1POLBSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640595-B1 SUBSTITUTED TERTIARY AMINO COMPOUND OR SALT THEREOF YAMANOUCHI PHARMA CO LTD (JP) 1999-03-24 EP disclosed
CN-1039228-C Novel substituted tert-amino compund YAMANOUCHI PHARMA CO LTD (JP) 1998-07-22 CN disclosed
US-5538976-A ANTICARCINOGENIC AGENTS AND ENZYME INHIBITORS FOR AROMATASE YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1996-07-23 US disclosed
EP-0640595-A1 NOVEL SUBSTITUTED TERTIARY AMINO COMPOUND OR SALT THEREOF YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1995-03-01 EP disclosed
CN-1079962-A New substituted tertiary amine compound and salt thereof YAMANOUCHI PHARMA CO LTD (JP) 1993-12-29 CN disclosed