SCHEMBL8327623

SCHEMBL8327623

O=[N+]([O-])c1ccc(N(Cc2ccc(Cl)cc2)c2cncnc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.50
CYP1A2 P05177 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
MAPT P10636 3/20 0.43
HTT P42858 3/20 0.43
NPC1 O15118 1/20 0.43
GAA P10253 1/20 0.43
RAB9A P51151 1/20 0.43
LMNA P02545 1/20 0.43
TP53 P04637 1/20 0.43
CRHBP P24387 2/20 0.42
CRHR2 Q13324 2/20 0.42
AR P10275 3/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
CYP19A1 P11511 2/20 0.41
NR1D1 P20393 1/20 0.41
NR1H3 Q13133 1/20 0.41
USP2 O75604 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8327952 0.93 CRHBP (0.47) ALDH1A1CYP1A2CYP2C9CYP2C19CRHBP
SCHEMBL8323939 0.87 AR (0.49) NPC1RAB9ACRHBPCRHR2AR
SCHEMBL8327171 0.87 CRHBP (0.42) ALDH1A1CYP1A2CYP2C9CYP2C19MAPT
SCHEMBL8326188 0.87 CYP19A1 (0.55) ALDH1A1MAPTHTTNPC1RAB9A
SCHEMBL8323517 0.84 KCNJ1 (0.46) MAPTNPC1CRHBPCRHR2AR
SCHEMBL8324619 0.84 KCNJ1 (0.46) MAPTNPC1CRHBPCRHR2AR
SCHEMBL8329070 0.84 MMP1 (0.45) MAPTRAB9ACRHBPCRHR2AR
SCHEMBL8329428 0.76 MAOA (0.42) CRHBPCRHR2CYP19A1NR1D1NR1H3
SCHEMBL3152135 0.72 PYCR1 (0.62) ALDH1A1CYP1A2CYP2C9CYP2C19MAPT
SCHEMBL5843018 0.72 CRHBP (0.64) ALDH1A1CYP1A2CYP2C9CYP2C19HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640595-B1 SUBSTITUTED TERTIARY AMINO COMPOUND OR SALT THEREOF YAMANOUCHI PHARMA CO LTD (JP) 1999-03-24 EP disclosed
US-5538976-A ANTICARCINOGENIC AGENTS AND ENZYME INHIBITORS FOR AROMATASE YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1996-07-23 US disclosed
EP-0640595-A1 NOVEL SUBSTITUTED TERTIARY AMINO COMPOUND OR SALT THEREOF YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1995-03-01 EP disclosed