SCHEMBL8324959

SCHEMBL8324959

CC(C)c1cccc([CH]C(Cc2ccccc2)N(C)C)c1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 4/20 0.39
SLC6A2 P23975 3/20 0.39
TAAR1 Q96RJ0 2/20 0.39
SLC6A4 P31645 2/20 0.39
SLC6A3 Q01959 2/20 0.39
MAOA P21397 1/20 0.39
CYP2A6 P11509 1/20 0.39
ADORA2A P29274 1/20 0.39
ADORA1 P30542 1/20 0.39
BACE1 P56817 3/20 0.38
BCHE P06276 10/20 0.38
ACHE P22303 8/20 0.38
ADRA2B P18089 1/20 0.37
ADRA2C P18825 1/20 0.37
HTR2A P28223 1/20 0.37
ADRA1A P35348 1/20 0.37
OPRK1 P41145 1/20 0.37
KCNH2 Q12809 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8324682 0.82 TP53 (0.40) SIGMAR1SLC6A2TAAR1SLC6A4SLC6A3
SCHEMBL8324358 0.82 TAAR1 (0.43) SIGMAR1SLC6A2TAAR1SLC6A4SLC6A3
SCHEMBL8327755 0.81 PNMT (0.41) SIGMAR1TAAR1
SCHEMBL8326976 0.81 MAOB (0.45) SIGMAR1SLC6A2TAAR1SLC6A4SLC6A3
SCHEMBL8324481 0.81 NFE2L2 (0.45) SIGMAR1SLC6A2TAAR1SLC6A4SLC6A3
SCHEMBL8322396 0.78 HTR2A (0.46) SIGMAR1SLC6A4ADRA2CHTR2AADRA1A
SCHEMBL8322028 0.77 TAAR1 (0.44) SIGMAR1SLC6A2TAAR1SLC6A4SLC6A3
SCHEMBL8325718 0.74 CYP2C19 (0.40) SIGMAR1SLC6A2TAAR1SLC6A4SLC6A3
SCHEMBL8323592 0.73 NOS3 (0.40) SIGMAR1SLC6A2SLC6A4SLC6A3MAOA
SCHEMBL8323270 0.72 KDM4E (0.36) SLC6A2SLC6A4SLC6A3ADRA2BADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0948496-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDONE COMPOUNDS AND METHODS OF USE Amgen inc. (US) 1999-10-13 EP disclosed
WO-1998024780-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDINONE COMPOUNDS AND THEIR USE AMGEN INC. (US) 1998-06-11 WO disclosed