SCHEMBL8325154

SCHEMBL8325154

O=C(O)[C@H]1C[C@H]2CCC[C@H]2N1S(=O)(=O)c1ccc(S(=O)(=O)c2ccccc2)s1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.42
MMP8 P22894 3/20 0.40
MMP12 P39900 1/20 0.40
MMP13 P45452 1/20 0.40
POLB P06746 1/20 0.40
ATM Q13315 1/20 0.37
LMNA P02545 2/20 0.37
TDP1 Q9NUW8 1/20 0.37
HTT P42858 1/20 0.37
ACHE P22303 1/20 0.36
NPC1 O15118 1/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
TSHR P16473 2/20 0.36
LOX P28300 3/20 0.36
LOXL2 Q9Y4K0 2/20 0.36
MAOA P21397 1/20 0.36
GAA P10253 1/20 0.35
HCRTR1 O43613 1/20 0.35
HCRTR2 O43614 1/20 0.35
MMP3 P08254 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13201305 0.82 MMP8 (0.60) ALDH1A1MMP8MMP12MMP13POLB
SCHEMBL7971275 0.81 ACHE (0.48) ALDH1A1ATMLMNATDP1HTT
SCHEMBL13201304 0.79 POLB (0.54) ALDH1A1POLBLMNATDP1HTT
SCHEMBL8319435 0.77 MMP2 (0.48) ALDH1A1MMP8MMP12ATMLMNA
SCHEMBL13201290 0.75 AKR1C3 (0.56) ALDH1A1LMNATDP1L3MBTL1TSHR
SCHEMBL8327363 0.75 MMP2 (0.48) ALDH1A1MMP8MMP12TDP1L3MBTL1
SCHEMBL13480182 0.74 KDM4E (0.48) ALDH1A1MMP8MMP12MMP13POLB
SCHEMBL8325166 0.74 KDM4E (0.48) ALDH1A1MMP8MMP12MMP13POLB
SCHEMBL8320725 0.73 EPHX2 (0.42) ALDH1A1ATMLMNATDP1HTT
SCHEMBL2964063 0.73 PSEN1 (0.43) ALDH1A1MMP12POLBATMLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7772270-B2 Imino acid derivatives as inhibitors of matrix metalloproteinases SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2010-08-10 US disclosed
US-7772270-B2 Imino acid derivatives as inhibitors of matrix metalloproteinases SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2010-08-10 US disclosed
EP-1585728-B1 IMINO ACID DERIVATIVES FOR USE AS INHIBITORS OF MATRIX METALLOPROTEINASES SANOFI AVENTIS DEUTSCHLAND (DE) 2010-02-24 EP disclosed