SCHEMBL8326665

SCHEMBL8326665

Cn1c(NC2CC3COCC(C2)N3Cc2ccc(F)cc2)c(C#N)c(=N)n(C)c1=S

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 1/20 0.34
MAPT P10636 2/20 0.34
OPRK1 P41145 1/20 0.34
DRD3 P35462 5/20 0.33
ALDH1A1 P00352 2/20 0.32
MITF O75030 1/20 0.32
HTT P42858 1/20 0.32
RAB9A P51151 1/20 0.32
KDM4E B2RXH2 1/20 0.31
HSD17B10 Q99714 1/20 0.31
DRD2 P14416 4/20 0.30
DRD4 P21917 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8887289 0.87 LTA4H (0.33) LTA4HMAPTOPRK1DRD3ALDH1A1
SCHEMBL8327067 0.87 LTA4H (0.33) LTA4HMAPTOPRK1DRD3ALDH1A1
SCHEMBL8325986 0.85 HRH1 (0.35) DRD3ALDH1A1HTTKDM4EDRD2
SCHEMBL8327922 0.83 BCHE (0.35) MAPTDRD3ALDH1A1MITFHTT
SCHEMBL8327173 0.81 PRKAA2 (0.42) DRD3ALDH1A1
SCHEMBL8326062 0.81 HTR3A (0.30)
SCHEMBL8328991 0.75 ALDH1A1 (0.31) MAPTALDH1A1MITFHTTRAB9A
SCHEMBL8322051 0.74 ALDH1A1 (0.42) MAPTALDH1A1MITFHTTRAB9A
SCHEMBL8324780 0.73
SCHEMBL8324755 0.73 SIGMAR1 (0.37) MAPTALDH1A1MITFHTTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0760368-B1 PYRIMIDINE DERIVATIVES NISSHIN FLOUR MILLING CO (JP) 1999-07-28 EP disclosed
US-5736550-A TREATMENT OF GASTROINTESTINAL TRACT DISORDERS NISSHIN FLOUR MILLING CO., LTD. (JP) 1998-04-07 US disclosed
EP-0760368-A1 NOVEL PYRIMIDINE DERIVATIVE NISSHIN FLOUR MILLING CO., LTD. (JP) 1997-03-05 EP disclosed