SCHEMBL8327173

SCHEMBL8327173

Cn1c(NC2CCN(Cc3ccc(F)cc3)CC2)c(C#N)c(=N)n(C)c1=S

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PRKAA2 P54646 4/20 0.42
ACHE P22303 5/20 0.42
BCHE P06276 2/20 0.42
BACE1 P56817 2/20 0.42
MCHR1 Q99705 2/20 0.40
SIGMAR1 Q99720 2/20 0.39
SSTR5 P35346 1/20 0.39
PRKAB2 O43741 2/20 0.39
PRKAG1 P54619 2/20 0.39
PRKAA1 Q13131 2/20 0.39
PRKAG3 Q9UGI9 2/20 0.39
PRKAG2 Q9UGJ0 2/20 0.39
PRKAB1 Q9Y478 2/20 0.39
CCNK O75909 1/20 0.38
CDK12 Q9NYV4 1/20 0.38
DRD3 P35462 1/20 0.38
ALDH1A1 P00352 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8327922 0.91 BCHE (0.35) PRKAA2ACHEBCHEBACE1PRKAB2
SCHEMBL8328374 0.87 ACHE (0.42) ACHE
SCHEMBL8324755 0.84 SIGMAR1 (0.37) ACHESIGMAR1ALDH1A1
SCHEMBL8328418 0.81 POLB (0.44) ALDH1A1
SCHEMBL8326665 0.81 LTA4H (0.34) DRD3ALDH1A1
SCHEMBL8328371 0.79 NOS3 (0.35)
SCHEMBL8326767 0.78 DRD4 (0.47) SIGMAR1DRD3
SCHEMBL8326437 0.78 KDM4E (0.43) ACHEDRD3
SCHEMBL8322051 0.77 ALDH1A1 (0.42) ALDH1A1
SCHEMBL8326581 0.77 SPHK2 (0.34) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0760368-B1 PYRIMIDINE DERIVATIVES NISSHIN FLOUR MILLING CO (JP) 1999-07-28 EP disclosed
US-5736550-A TREATMENT OF GASTROINTESTINAL TRACT DISORDERS NISSHIN FLOUR MILLING CO., LTD. (JP) 1998-04-07 US disclosed
EP-0760368-A1 NOVEL PYRIMIDINE DERIVATIVE NISSHIN FLOUR MILLING CO., LTD. (JP) 1997-03-05 EP disclosed