SCHEMBL8326774

SCHEMBL8326774

CNC([CH]c1ccc(C(F)(F)F)cc1)Cc1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.52
RAB9A P51151 3/20 0.52
NOS3 P29474 1/20 0.46
NOS1 P29475 1/20 0.46
NOS2 P35228 1/20 0.46
PPARG P37231 1/20 0.42
PPARA Q07869 1/20 0.42
FPR2 P25090 1/20 0.41
TAAR1 Q96RJ0 2/20 0.41
SIGMAR1 Q99720 2/20 0.41
SLC18A2 Q05940 1/20 0.41
MAPT P10636 2/20 0.40
TP53 P04637 2/20 0.40
POLB P06746 1/20 0.40
CNR2 P34972 1/20 0.39
CTSL P07711 1/20 0.39
LMNA P02545 2/20 0.39
MAPK1 P28482 2/20 0.39
GRIN2B Q13224 2/20 0.38
MTOR P42345 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8326920 0.85 HTR2A (0.46) NPC1RAB9APPARGPPARASIGMAR1
SCHEMBL8324972 0.83 TAAR1 (0.44) NOS3NOS1NOS2PPARGPPARA
SCHEMBL8325444 0.81 TAAR1 (0.46) PPARGPPARATAAR1SIGMAR1SLC18A2
SCHEMBL8326251 0.80 NPC1 (0.59) NPC1RAB9ANOS3NOS1NOS2
SCHEMBL8323399 0.78 LTA4H (0.50) PPARGPPARAFPR2TAAR1SIGMAR1
SCHEMBL8322987 0.77 NPC1 (0.52) NPC1RAB9ANOS3NOS1NOS2
SCHEMBL8322850 0.73 NFE2L2 (0.45) NPC1RAB9APPARGPPARATAAR1
SCHEMBL8322029 0.73 CYP3A4 (0.40) NPC1RAB9ANOS2PPARGPPARA
SCHEMBL8327429 0.72 TAAR1 (0.42) NPC1TAAR1SIGMAR1SLC18A2TP53
SCHEMBL8325015 0.71 MAOA (0.45) TAAR1SIGMAR1SLC18A2MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0948496-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDONE COMPOUNDS AND METHODS OF USE Amgen inc. (US) 1999-10-13 EP disclosed
WO-1998024780-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDINONE COMPOUNDS AND THEIR USE AMGEN INC. (US) 1998-06-11 WO disclosed