SCHEMBL8328585

SCHEMBL8328585

CN(CCC1CCCCN1Cc1ccc(F)cc1)c1c(C#N)c(=N)n(C)c(=S)n1C

nearest known ligand 0.34

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.34
KDM4E B2RXH2 1/20 0.34
SLC6A4 P31645 2/20 0.33
SPHK2 Q9NRA0 2/20 0.33
SPHK1 Q9NYA1 2/20 0.33
NPSR1 Q6W5P4 1/20 0.32
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
OPRK1 P41145 1/20 0.31
SIGMAR1 Q99720 1/20 0.30
MAPK1 P28482 1/20 0.30
RORC P51449 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8326577 0.84 ALDH1A1 (0.34) ALDH1A1KDM4ENPSR1SIGMAR1
SCHEMBL8326581 0.80 SPHK2 (0.34) ALDH1A1SPHK2SPHK1NPSR1MAPK1
SCHEMBL8328415 0.76 GSK3B (0.36) MEN1KMT2ASIGMAR1
SCHEMBL8328371 0.75 NOS3 (0.35)
SCHEMBL8328988 0.74 KDM4E (0.31) ALDH1A1KDM4EMEN1KMT2A
SCHEMBL8326763 0.72 DRD4 (0.41) ALDH1A1KDM4E
SCHEMBL8617181 0.69 ALDH1A1 (0.35) ALDH1A1KDM4ENPSR1MEN1KMT2A
SCHEMBL8327665 0.69 ALDH1A1 (0.39) ALDH1A1KDM4ESLC6A4SPHK2SPHK1
SCHEMBL8327662 0.69 KDM4E (0.39) ALDH1A1KDM4ESLC6A4SPHK2SPHK1
SCHEMBL8328991 0.68 ALDH1A1 (0.31) ALDH1A1KDM4ESIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0760368-B1 PYRIMIDINE DERIVATIVES NISSHIN FLOUR MILLING CO (JP) 1999-07-28 EP disclosed
EP-0760368-A1 NOVEL PYRIMIDINE DERIVATIVE NISSHIN FLOUR MILLING CO., LTD. (JP) 1997-03-05 EP disclosed