SCHEMBL8326581

SCHEMBL8326581

Cn1c(NCC2CCCCN2Cc2ccc(F)cc2)c(C#N)c(=N)n(C)c1=S

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SPHK2 Q9NRA0 2/20 0.34
SPHK1 Q9NYA1 2/20 0.34
OPRM1 P35372 1/20 0.34
ALDH1A1 P00352 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
LMNA P02545 1/20 0.32
HDAC8 Q9BY41 2/20 0.32
HDAC6 Q9UBN7 2/20 0.32
HDAC1 Q13547 1/20 0.32
MAPK1 P28482 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8328991 0.85 ALDH1A1 (0.31) ALDH1A1LMNA
SCHEMBL8328374 0.82 ACHE (0.42)
SCHEMBL8328418 0.81 POLB (0.44) ALDH1A1LMNA
SCHEMBL8328585 0.80 ALDH1A1 (0.34) SPHK2SPHK1ALDH1A1NPSR1MAPK1
SCHEMBL8326577 0.78 ALDH1A1 (0.34) ALDH1A1NPSR1
SCHEMBL8326767 0.77 DRD4 (0.47) LMNA
SCHEMBL8327173 0.77 PRKAA2 (0.42) ALDH1A1
SCHEMBL8324755 0.77 SIGMAR1 (0.37) ALDH1A1MAPK1
SCHEMBL8322051 0.76 ALDH1A1 (0.42) ALDH1A1MAPK1
SCHEMBL8327922 0.75 BCHE (0.35) ALDH1A1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0760368-B1 PYRIMIDINE DERIVATIVES NISSHIN FLOUR MILLING CO (JP) 1999-07-28 EP disclosed
US-5736550-A TREATMENT OF GASTROINTESTINAL TRACT DISORDERS NISSHIN FLOUR MILLING CO., LTD. (JP) 1998-04-07 US disclosed
EP-0760368-A1 NOVEL PYRIMIDINE DERIVATIVE NISSHIN FLOUR MILLING CO., LTD. (JP) 1997-03-05 EP disclosed