SCHEMBL8347291

SCHEMBL8347291

COc1ccc([C]2CCNC2)cc1OC

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 3/20 0.46
PDE4B Q07343 3/20 0.45
PDE4C Q08493 2/20 0.45
PDE4D Q08499 2/20 0.45
PDE3B Q13370 1/20 0.45
PDE3A Q14432 1/20 0.45
QDPR P09417 1/20 0.44
ALDH1A1 P00352 3/20 0.44
KDM4E B2RXH2 2/20 0.44
MAPT P10636 1/20 0.44
THRB P10828 1/20 0.44
TLR9 Q9NR96 2/20 0.42
TLR7 Q9NYK1 2/20 0.42
CD274 Q9NZQ7 1/20 0.42
TDP1 Q9NUW8 2/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
GAA P10253 1/20 0.41
MPI P34949 1/20 0.41
GFER P55789 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8640742 0.87 PTGS2 (0.44) QDPRCD274
SCHEMBL9869903 0.78 PDE4A (0.57) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL8638940 0.78 NISCH (0.43) THRBCD274TSHRHSD17B10
SCHEMBL7305529 0.75 QDPR (0.76) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL11198805 0.75 ADRA2A (0.55) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL8640758 0.74 HTR7 (0.41) MAPTCD274
SCHEMBL10819033 0.74 SOS1 (0.59) PDE4APDE4BPDE4CPDE4DNPC1
SCHEMBL8840880 0.73 PDE4A (0.67) PDE4AALDH1A1KDM4EMAPTTHRB
SCHEMBL27582163 0.73 PDE4A (0.52) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL8350829 0.70 AHR (0.48) ALDH1A1KDM4EMAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5861416-A TREATMENT OF ASTHMA OR COUGH MERRELL PHARMACEUTICALS INC. (US) 1999-01-19 US disclosed
US-5824690-A TREATING ASTHMA, COUGH HOECHST MARION ROUSSEL INC. (US) 1998-10-20 US disclosed