SCHEMBL8350829

SCHEMBL8350829

Clc1ccc([C]2CCNC2)cc1Cl

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AHR P35869 5/20 0.48
SLC6A2 P23975 2/20 0.46
SLC6A4 P31645 2/20 0.46
SLC6A3 Q01959 2/20 0.46
CYP1B1 Q16678 1/20 0.42
PNMT P11086 6/20 0.42
ADRA2A P08913 1/20 0.42
ADRA2B P18089 1/20 0.42
ADRA2C P18825 1/20 0.42
ASIC3 Q9UHC3 1/20 0.41
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
HTR2B P41595 1/20 0.40
MAPT P10636 2/20 0.39
HTT P42858 2/20 0.39
ALDH1A1 P00352 1/20 0.39
HPGD P15428 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
NOTUM Q6P988 1/20 0.38
KDM4E B2RXH2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27997002 0.88 AHR (0.52) AHRSLC6A2SLC6A4SLC6A3CYP1B1
SCHEMBL8640742 0.80 PTGS2 (0.44) HTR2AHTR2CHTR2BMEN1KMT2A
SCHEMBL8638141 0.78 SIGMAR1 (0.52) PNMTADRA2AADRA2BADRA2CASIC3
SCHEMBL9870874 0.77 AHR (0.65) AHRSLC6A2SLC6A3CYP1B1MAPT
SCHEMBL8639724 0.76 HTR2C (0.56) SLC6A4PNMTASIC3HTR2AHTR2C
SCHEMBL8640758 0.73 HTR7 (0.41) PNMTASIC3MAPTNOTUMUSP2
SCHEMBL8638170 0.73 MLNR (0.39) PNMTASIC3HTR2AHTR2CHTR2B
SCHEMBL6472818 0.73 AHR (0.59) AHRSLC6A2SLC6A4SLC6A3CYP1B1
SCHEMBL4808905 0.71 AHR (0.56) AHRSLC6A2SLC6A3CYP1B1MAPT
SCHEMBL30022165 0.70 ADRA2A (0.60) AHRSLC6A2SLC6A4SLC6A3CYP1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5861416-A TREATMENT OF ASTHMA OR COUGH MERRELL PHARMACEUTICALS INC. (US) 1999-01-19 US disclosed
US-5824690-A TREATING ASTHMA, COUGH HOECHST MARION ROUSSEL INC. (US) 1998-10-20 US disclosed