Phenethylamine

Phenethylamine

SCHEMBL8384113

NCCc1ccccc1.O

nearest known ligand 0.94

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABCC9ABL1ACEACHEACVR1ADORA1ADORA2AADORA2BADORA3ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALOX5ATP4AATP4BBCRBTKCACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGCRBNCUL4ACXCR1CXCR2DDB1DDCDHFRDPP4DRD2DRD3DRD4EGFRERBB2ERBB4ESR1ESR2FDPSFKBP1AFLT1FLT3FLT4GARTGHSRGRIA1GRIA2GRIA3GRIA4GRIK1GRIK2GRIK3GRIK4GRIK5GRIN2AGSK3AGSK3BHDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IDH1IDH2IMPA1ITGA2BITGB3JAK1JAK2JAK3KCNJ11KCNK3KCNK9KDRKITMEN1METMMP1MMP13MMP7MMP8NANOD2NS5bODC1OPG057OPRD1OPRK1OPRM1PPARP1PARP2PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PKLRPPARDPPATPTGS1PTGS2RBX1ROCK1ROCK2RRM1RRM2RRM2BSCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC10A2SLC5A2SLC6A2SLC6A3SLC6A4SLC9A3SYKTACR1THRATHRBTOP1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYK2TYMSVDRampCblablaT-3blaT-4blaT-5blaT-6blaUOE-1dacAdacBdacCfolAfolPftsIgyrAgyrBileSmecAmrcAmrcBmrdAparCparEpbp2pbp4pbpApbpFrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUthyAykgMykgO

The experimentally established mechanism targets of Phenethylamine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR2A known ✓ P28223 3/20 0.94
HTR6 known ✓ P50406 2/20 0.56
HTR2C known ✓ P28335 1/20 0.54
LOXL2 Q9Y4K0 2/20 0.94
TAAR1 Q96RJ0 2/20 0.94
CYP2A6 P11509 1/20 0.94
SMN1; SMN2 Q16637 1/20 0.94
MAOA P21397 3/20 0.64
MAOB P27338 3/20 0.59
CYP1A2 P05177 1/20 0.58
CYP2D6 P10635 1/20 0.58
CYP2C19 P33261 1/20 0.58
ALDH1A1 P00352 1/20 0.52
HPGD P15428 1/20 0.52
ALOX15 P16050 1/20 0.52
ALOX12 P18054 1/20 0.52
CASP1 P29466 1/20 0.52
HSD17B10 Q99714 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Phenethylamine SCHEMBL1331271 0.97
Phenethylamine SCHEMBL1330939 0.97
Phenethylamine SCHEMBL27634208 0.97 HTR2A (1.00) HTR2ALOXL2TAAR1CYP2A6SMN1; SMN2
Phenethylamine SCHEMBL1799333 0.97 HTR2A (1.00) HTR2ALOXL2TAAR1CYP2A6SMN1; SMN2
Phenethylamine SCHEMBL968 0.97
Phenethylamine SCHEMBL1332244 0.97
Phenethylamine SCHEMBL245154 0.94 HTR2A (0.94) HTR2ALOXL2TAAR1CYP2A6SMN1; SMN2
Phenethylamine SCHEMBL20568335 0.94 HTR2A (0.94) HTR2ALOXL2TAAR1CYP2A6SMN1; SMN2
Phenethylamine SCHEMBL10592571 0.94 HTR2A (0.94) HTR2ALOXL2TAAR1CYP2A6SMN1; SMN2
Phenethylamine SCHEMBL837569 0.94 HTR2A (0.94) HTR2ALOXL2TAAR1CYP2A6SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 46 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11024462-B2 Ceramic electronic component and method of manufacturing the same and electronic device SAMSUNG ELECTRONICS CO., LTD. (KR) 2021-06-01 US claimed
US-20200234888-A1 CERAMIC ELECTRONIC COMPONENT AND METHOD OF MANUFACTURING THE SAME AND ELECTRONIC DEVICE SAMSUNG ELECTRONICS CO LTD (KR) 2020-07-23 US claimed
US-20190131077-A1 CERAMIC ELECTRONIC COMPONENT AND METHOD OF MANUFACTURING THE SAME AND ELECTRONIC DEVICE NATIONAL INSTITUTE FOR MATERIALS SCIENCE (JP) 2019-05-02 US claimed
US-11763989-B2 Dielectric monolayer thin film, capacitor and semiconductor device each including the same, and method of forming the dielectric monolayer thin film SAMSUNG ELECTRONICS CO., LTD. (KR) 2023-09-19 US disclosed
US-11664414-B2 Single crystal material and method of forming the same and stacked structure and ceramic electronic component and device SAMSUNG ELECTRONICS CO., LTD. (KR) 2023-05-30 US disclosed
CN-110246689-B Ceramic dielectric and method for manufacturing the same, ceramic electronic component and electronic device 三星电子株式会社 2022-05-24 CN disclosed
US-11120944-B2 Ceramic electronic component including ceramic nanosheets having multimodal lateral size distribution and method of manufacturing the same and electronic device SAMSUNG ELECTRONICS CO., LTD. (KR) 2021-09-14 US disclosed
US-11024462-B2 Ceramic electronic component and method of manufacturing the same and electronic device SAMSUNG ELECTRONICS CO., LTD. (KR) 2021-06-01 US disclosed
US-20210134941-A1 SINGLE CRYSTAL MATERIAL AND METHOD OF FORMING THE SAME AND STACKED STRUCTURE AND CERAMIC ELECTRONIC COMPONENT AND DEVICE SAMSUNG ELECTRONICS CO LTD (KR) 2021-05-06 US disclosed
US-10993320-B2 Population of metal oxide nanosheets, preparation method thereof, and electrical conductor and electronic device including the same SAMSUNG ELECTRONICS CO., LTD. (KR) 2021-04-27 US disclosed
US-20210110975-A1 DIELECTRIC MONOLAYER THIN FILM, CAPACITOR AND SEMICONDUCTOR DEVICE EACH INCLUDING THE SAME, AND METHOD OF FORMING THE DIELECTRIC MONOLAYER THIN FILM SAMSUNG ELECTRONICS CO., LTD. (KR) 2021-04-15 US disclosed
US-5025034-A Thromboxane inhibitors NATIONAL RESEARCH DEVELOPMENT CORPORATION (GB) 1991-06-18 US disclosed
US-4945106-A Prostaglandins NATIONAL RESEARCH DEVELOPMENT CORPORATION (GB) 1990-07-31 US disclosed
EP-0111955-B1 PROSTAGLANDIN INTERMEDIATES NATIONAL RESEARCH DEVELOPMENT CORPORATION (GB) 1986-09-17 EP disclosed
US-4596823-A Prostaglandins NATIONAL RESEARCH DEVELOPMENT CORPORATION (GB) 1986-06-24 US disclosed
EP-0043292-B1 PROSTAGLANDINS NATIONAL RESEARCH DEVELOPMENT CORPORATION (GB) 1986-01-15 EP disclosed
EP-0142322-A2 Cyclohexane derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1985-05-22 EP disclosed
EP-0142323-A2 Process for making erythro-dihydroxyalkenoic acide derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1985-05-22 EP disclosed
WO-1982000142-A1 PROSTAGLANDINS JONES R 1982-01-21 WO disclosed
US-4130565-A 3-ALKYL-TETRAHYDROPYRAN-OR THIOPYRAN-2,4-DIONES AS CHEMICAL INTERMEDIATES SHIONOGI & CO., LTD. (JP) 1978-12-19 US disclosed