SCHEMBL838467

SCHEMBL838467

COC(=O)Cc1c(F)cccc1Cl

nearest known ligand 0.74

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.74
LMNA P02545 2/20 0.57
KMT2A Q03164 3/20 0.56
MEN1 O00255 2/20 0.56
TP53 P04637 1/20 0.55
MAPT P10636 1/20 0.54
NPC1 O15118 1/20 0.53
RAB9A P51151 1/20 0.53
ALDH1A1 P00352 2/20 0.53
HPGD P15428 1/20 0.53
POLB P06746 1/20 0.53
KDM4E B2RXH2 2/20 0.53
TSHR P16473 1/20 0.53
RXFP1 Q9HBX9 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3743731 0.88 AKR1B1 (0.59) SMN1; SMN2LMNAKMT2AMEN1MAPT
SCHEMBL9985451 0.88 SMN1; SMN2 (0.56) SMN1; SMN2LMNAKMT2AMEN1TP53
SCHEMBL5252336 0.84 KMT2A (0.60) SMN1; SMN2LMNAKMT2AMEN1MAPT
SCHEMBL7638563 0.84 SMN1; SMN2 (0.62) SMN1; SMN2LMNAKMT2AMEN1TP53
SCHEMBL29943508 0.84 KMT2A (0.60) SMN1; SMN2LMNAKMT2AMEN1MAPT
SCHEMBL28724963 0.81 SMN1; SMN2 (0.51) SMN1; SMN2LMNAKMT2AMEN1TP53
SCHEMBL28158406 0.81 SMN1; SMN2 (0.51) SMN1; SMN2KMT2AALDH1A1HPGDPOLB
SCHEMBL9729592 0.81 SMN1; SMN2 (0.58) SMN1; SMN2LMNAKMT2ATP53MAPT
SCHEMBL2373994 0.81 SMN1; SMN2 (0.51) SMN1; SMN2KMT2AALDH1A1HPGDKDM4E
SCHEMBL28031637 0.81 SMN1; SMN2 (0.51) SMN1; SMN2LMNAKMT2AMEN1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 27 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250163039-A1 HETEROAROMATIC COMPOUNDS FOR THE TREATMENT OF CANCER BOEHRINGER INGELHEIM INT (DE) 2025-05-22 US disclosed
EP-4452964-A1 HETEROAROMATIC COMPOUNDS FOR THE TREATMENT OF CANCER Boehringer Ingelheim International GmbH (DE) 2024-10-30 EP disclosed
CN-118339153-A Heteroaromatic compounds for the treatment of cancer 勃林格殷格翰国际有限公司 2024-07-12 CN disclosed
CN-116804004-A Compounds as DHODH inhibitors 南京征祥医药有限公司 2023-09-26 CN disclosed
US-20230271943-A1 COMPOUNDS AS DHODH INHIBITORS NANJING ZENSHINE PHARMACEUTICALS CO., LTD. (CN) 2023-08-31 US disclosed
US-20230271943-A1 COMPOUNDS AS DHODH INHIBITORS NANJING ZENSHINE PHARMACEUTICALS CO., LTD. (CN) 2023-08-31 US disclosed
CN-116457343-A Compounds as DHODH inhibitors 南京征祥医药有限公司 2023-07-18 CN disclosed
WO-2023117681-A1 HETEROAROMATIC COMPOUNDS FOR THE TREATMENT OF CANCER BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2023-06-29 WO disclosed
WO-2022012548-A1 COMPOUNDS AS DHODH INHIBITORS NANJING ZHENGXIANG PHARMACEUTICALS CO., LTD. (CN) 2022-01-20 WO disclosed
US-9738642-B2 Triazolopyridine ether derivatives and their use in neurological and pyschiatric disorders BRISTOL-MYERS SQUIBB COMPANY (US) 2017-08-22 US disclosed
US-8143280-B2 Glucocorticoid receptor antagonists HOFFMANN-LA ROCHE INC. (US) 2012-03-27 US disclosed
EP-2205562-B1 1,1,1-TRIFLUORO-2-HYDROXY-3-PHENYLPROPANE DERIVATIVES HOFFMANN LA ROCHE (CH) 2011-03-16 EP disclosed
CN-101808992-A 1,1,1-trifluoro-2-hydroxy-3-phenylpropane derivatives HOFFMANN LA ROCHE 2010-08-18 CN disclosed
EP-2205562-A1 1,1,1-TRIFLUORO-2-HYDROXY-3-PHENYLPROPANE DERIVATIVES F. Hoffmann-Roche AG (CH) 2010-07-14 EP disclosed
US-20090088425-A1 GLUCOCORTICOID RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2009-04-02 US disclosed
WO-2009040288-A1 1,1,1-TRIFLUORO-2-HYDROXY-3-PHENYLPROPANE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2009-04-02 WO disclosed
WO-2003076403-A1 1,2-DISUBSTITUDED-6-OXO-3-PHENYL-PIPERIDINE-3-CARBOXAMIDES AND COMBINATORIAL LIBRARIES THEREOF LION BIOSCIENCE AG (DE) 2003-09-18 WO disclosed
US-20030171588-A1 1,2-disubstituted-6-oxo-3-phenyl-piperidine-3-carboxamides and combinatorial libraries thereof LION BIOSCIENCE AG (DE) 2003-09-11 US disclosed
CN-1008055-B PESTICIDE COMPOSITION WITH ACRYLIC DERIVS. AS ACTIVE COMPONENT AND PROCESS FOR PREPARING SAME, AND USE THEREOF ICI PLC (GB) 1990-05-23 CN disclosed
CN-85108235-A The preparation of sterilant 1986-08-27 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030171588-A1 1,2-disubstituted-6-oxo-3-phenyl-piperidine-3-carboxamides and combinatorial libraries thereof BRD4, BICRA, HDAC6 SMN1; SMN2 1499/4885LMNA 3593/4885KMT2A 202/4885
US-20250163039-A1 HETEROAROMATIC COMPOUNDS FOR THE TREATMENT OF CANCER NRAS, KRAS, RB1 SMN1; SMN2 4332/4885LMNA 2852/4885KMT2A 2424/4885
US-20230271943-A1 COMPOUNDS AS DHODH INHIBITORS DHODH, DLD, DHRS9 SMN1; SMN2 3538/4885LMNA 3421/4885KMT2A 2940/4885
US-20090088425-A1 GLUCOCORTICOID RECEPTOR ANTAGONISTS NR3C1, NR3C2, MC2R SMN1; SMN2 4680/4885LMNA 2031/4885KMT2A 2149/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.