SCHEMBL8416993

SCHEMBL8416993

COC(=O)C(C#N)Cc1ccc(N=C=O)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.44
TSHR P16473 1/20 0.44
ANPEP P15144 4/20 0.40
ESR1 P03372 1/20 0.38
ESR2 Q92731 1/20 0.38
PLG P00747 6/20 0.37
PLAU P00749 6/20 0.37
F2 P00734 5/20 0.37
PLAT P00750 5/20 0.37
MAPK1 P28482 1/20 0.37
MIF P14174 1/20 0.36
PTPRB P23467 1/20 0.35
CYP1A2 P05177 1/20 0.35
F10 P00742 2/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
NLRP3 Q96P20 1/20 0.33
KLK8 O60259 1/20 0.33
KLK2 P20151 1/20 0.33
KLK4 Q9Y5K2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL433224 0.81 ESR1 (0.58) CYP3A4TSHRANPEPESR1ESR2
SCHEMBL28384249 0.81 ATM (0.46) ANPEPESR1ESR2MAPK1MIF
SCHEMBL31474258 0.80 NOS2 (0.48) TSHRANPEPESR1ESR2MAPK1
SCHEMBL11925791 0.80 NLRP3 (0.47) CYP3A4ANPEPESR1ESR2MAPK1
SCHEMBL12321430 0.80 CTSC (0.49) ANPEPESR1ESR2MAPK1KMT2A
SCHEMBL10523997 0.79 ANPEP (0.57) ANPEPMEN1KMT2A
SCHEMBL11924843 0.79 MIF (0.46) CYP3A4TSHRANPEPESR1ESR2
SCHEMBL9788997 0.78 TAS1R3 (0.46) ANPEPESR1ESR2MAPK1
SCHEMBL21763387 0.77 ANPEP (0.52) CYP3A4ANPEPCYP1A2
SCHEMBL10536462 0.77 ALDH1A1 (0.47) TSHRANPEPESR1ESR2MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5880284-A HAVING ANTITHROMBOTIC, ANTIAGGREGATORY AND TUMOR- OR METASTASES-INHIBITING EFFECTS DR. KARL THOMAE GMBH (DE) 1999-03-09 US disclosed
US-5681841-A PREVENTION CELL AGGREGATION KARL THOMAE GMBH (DE) 1997-10-28 US disclosed