SCHEMBL8427341

SCHEMBL8427341

COCc1ccc2c(N3C(=O)C=C(c4cn(C)c5ccccc45)C3=O)cn(C(C)C)c2c1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CCNT1 O60563 4/20 0.42
CDK9 P50750 4/20 0.42
CDK2 P24941 2/20 0.42
CCNA2 P20248 1/20 0.42
PTPRC P08575 1/20 0.39
GSK3B P49841 5/20 0.38
PRKCA P17252 6/20 0.34
PRKCB P05771 2/20 0.34
PRKCH P24723 1/20 0.34
PRKCE Q02156 1/20 0.34
PRKCQ Q04759 1/20 0.34
PRKCD Q05655 1/20 0.34
CCNE2 O96020 1/20 0.33
CDK4 P11802 1/20 0.33
CCND1 P24385 1/20 0.33
CCNE1 P24864 1/20 0.33
KDR P35968 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6950830 0.78 CCNE2 (0.58) CDK2GSK3BPRKCAPRKCBPRKCH
SCHEMBL8466339 0.71 CCNT1 (0.44) CCNT1CDK9CDK2CCNA2PTPRC
SCHEMBL8619764 0.70 CAMK2D (0.57) CCNT1CDK9CDK2CCNA2PTPRC
SCHEMBL8920747 0.70 PRKCG (0.61) CCNT1CDK9CDK2CCNA2PTPRC
SCHEMBL6945284 0.69 CCNE2 (0.67) CDK2GSK3BPRKCAPRKCBPRKCH
SCHEMBL5957039 0.69 GSK3B (0.53) CCNT1CDK9CDK2CCNA2PTPRC
SCHEMBL29447190 0.69 GSK3B (0.53) CCNT1CDK9CDK2CCNA2PTPRC
SCHEMBL25282614 0.68 CAMK2D (0.57) CCNT1CDK9CDK2CCNA2
SCHEMBL8923158 0.68 GSK3B (0.47) CCNT1CDK9CDK2CCNA2GSK3B
SCHEMBL8477960 0.67 CCNT1 (0.42) CCNT1CDK9CDK2CCNA2PTPRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5856517-A ANTIPROLIFERATIVE AGENTS USEFUL IN THE TREATMENT OF CANCER. HOFFMANN-LA ROCHE INC. (US) 1999-01-05 US disclosed