SCHEMBL8429155

SCHEMBL8429155

O=CNN([C@@H](Cc1ccccc1)C(=O)Oc1cccc(NC2=NCCN2)c1)S(=O)(=O)c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 11/20 0.46
ITGAV P06756 11/20 0.46
ITGA2B P08514 8/20 0.46
ITGB1 P05556 2/20 0.42
ITGB5 P18084 2/20 0.42
PTGIR P43119 5/20 0.38
F2 P00734 1/20 0.35
C1R P00736 1/20 0.35
F10 P00742 1/20 0.35
KLKB1 P03952 1/20 0.35
KLK1 P06870 1/20 0.35
PRSS1 P07477 1/20 0.35
ADRA2A P08913 1/20 0.34
GPR65 Q8IYL9 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8430878 0.80 CA12 (0.39)
SCHEMBL8431123 0.79 ITGB3 (0.54) ITGB3ITGAVITGA2BITGB1ITGB5
SCHEMBL8429288 0.71 CA2 (0.38) F2KLKB1PRSS1
SCHEMBL8432878 0.70 ITGB3 (0.39) ITGB3ITGAVITGA2B
SCHEMBL8432271 0.70 ACHE (0.33) ITGB3ITGAVITGA2BITGB1ITGB5
SCHEMBL8429051 0.68 SIRT2 (0.36) F2F10PRSS1
SCHEMBL8431173 0.67 CTSD (0.35) F2KLKB1PRSS1
SCHEMBL11168815 0.66 ADRA2A (0.66) PTGIRADRA2A
SCHEMBL7863191 0.65 KMT2A (0.47) ITGB3ITGAVITGA2BITGB1ITGB5
Hydrochloric Acid SCHEMBL11160123 0.65 ADRA2A (0.64) PTGIRADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5952381-A SELECTIVELY INHIBITING OR ANTAGONIZING THE INTEGRINS; ANTITUMOR AGENTS, ANTIARTHRITIC AGENTS, VIRICIDES, MICROBIOCIDES; TREATING OSTEOPOROSIS, SKIN DISORDERS G. D. SEARLE & CO. (US) 1999-09-14 US disclosed