SCHEMBL8433448

SCHEMBL8433448

CN(C)CC1CCc2ccc(NC=O)cc21

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 5/20 0.43
ADRA2A P08913 1/20 0.40
ADRA2B P18089 1/20 0.40
ADRA2C P18825 1/20 0.40
ADRA1D P25100 1/20 0.40
ADRA1A P35348 1/20 0.40
ADRA1B P35368 1/20 0.40
HTR6 P50406 1/20 0.37
NQO2 P16083 3/20 0.36
MTNR1B P49286 3/20 0.36
OPRD1 P41143 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8436848 0.85 ADRA2A (0.44) MTNR1AADRA2AADRA2BADRA2CADRA1D
SCHEMBL8521222 0.82 ADRA2A (0.46) MTNR1AADRA2AADRA2BADRA2CADRA1D
SCHEMBL8433848 0.80 MTNR1A (0.67) MTNR1ANQO2MTNR1B
Oxalic Acid SCHEMBL8432164 0.80 ADRA2A (0.43) MTNR1AADRA2AADRA2BADRA2CADRA1D
SCHEMBL8432229 0.76 MTNR1A (0.39) MTNR1AOPRD1
SCHEMBL8432175 0.75 MTNR1A (0.39) MTNR1AOPRD1
Dimethylamine SCHEMBL8433452 0.74 OPRD1 (0.38) MTNR1AADRA2AADRA2BADRA2COPRD1
SCHEMBL9628347 0.74 ESR1 (0.60) MTNR1AADRA2AADRA2BADRA2CADRA1D
SCHEMBL7101452 0.74 ACHE (0.42) MTNR1AOPRD1
SCHEMBL7950364 0.73 MTNR1A (0.41) MTNR1AHTR6NQO2MTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5972964-A FOR TREATMENT OF CERTAIN PSYCHIC AND NEUROLOGIC DISORDERS SUCH AS PSYCHOSIS, ANXIETY DISORDERS, PANIC DISORDER, OBSESSIVE COMPULSIVE DISORDER, DEPRESSION, IMPULSE CONTROL DISORDERS, ALCOHOL ABUSE, AGGRESSION H. LUNDBECK A/S (DK) 1999-10-26 US disclosed
US-5807889-A PSYCHOLOGICAL AND NERVOUS SYSTEM DISORDERS H. LUNDBECK A/S (DK) 1998-09-15 US disclosed
EP-0673360-B1 AMINOMETHYLINDANS, -BENZOFURANES AND -BENZOTHIOPHENES LUNDBECK & CO AS H (DK) 1998-08-26 EP disclosed
EP-0673360-A1 AMINOMETHYLINDANS, -BENZOFURANES AND -BENZOTHIOPHENES H. LUNDBECK A/S (DK) 1995-09-27 EP disclosed
WO-1994013620-A1 AMINOMETHYLINDANS, -BENZOFURANES AND -BENZOTHIOPHENES H. LUNDBECK A/S (DK) 1994-06-23 WO disclosed