SCHEMBL8444243

SCHEMBL8444243

CCN(CC)CCNS(=O)(=O)c1ccc(Oc2ccc(C(=O)NC(=N)N)cc2S(C)(=O)=O)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.53
MAPK1 P28482 1/20 0.53
GFER P55789 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.48
KMT2A Q03164 1/20 0.44
SIGMAR1 Q99720 2/20 0.43
USP2 O75604 1/20 0.41
LMNA P02545 2/20 0.41
CYP2C9 P11712 2/20 0.41
ADRA2A P08913 1/20 0.41
CYP2D6 P10635 1/20 0.41
DRD2 P14416 1/20 0.41
TSHR P16473 1/20 0.41
DRD3 P35462 1/20 0.41
HTR2B P41595 1/20 0.41
STAT6 P42226 1/20 0.41
KCNH2 Q12809 1/20 0.41
BLM P54132 1/20 0.41
OPRM1 P35372 1/20 0.39
OPRK1 P41145 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8070683 0.99 ALDH1A1 (0.52) ALDH1A1MAPK1GFERSMN1; SMN2KMT2A
SCHEMBL8068849 0.86 ALDH1A1 (0.54) ALDH1A1MAPK1GFERSMN1; SMN2KMT2A
SCHEMBL8444240 0.82 MRGPRX1 (0.37) ALDH1A1LMNA
SCHEMBL8444776 0.82 SIGMAR1 (0.46) ALDH1A1SMN1; SMN2KMT2ASIGMAR1USP2
Hydrochloric Acid SCHEMBL8070680 0.82 MRGPRX1 (0.36) ALDH1A1LMNA
SCHEMBL8068683 0.82 SMN1; SMN2 (0.41) SMN1; SMN2LMNATSHR
Hydrochloric Acid SCHEMBL8068487 0.81 SIGMAR1 (0.45) ALDH1A1SMN1; SMN2KMT2ASIGMAR1USP2
SCHEMBL8446348 0.81 CA2 (0.43) ALDH1A1KMT2ATSHRCA9
Hydrochloric Acid SCHEMBL8059609 0.81 SMN1; SMN2 (0.40) SMN1; SMN2LMNATSHR
SCHEMBL8446065 0.81 CYP19A1 (0.50) ALDH1A1SMN1; SMN2KMT2ATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0723956-B1 Basically substituted benzoylguanidines, process for their preparation, their use as medicaments or diagnostics as well as medicaments containing them HOECHST AG (DE) 1999-10-13 EP claimed