SCHEMBL845267

SCHEMBL845267

O=C(Nc1ccc(/C=C/c2ccc(NC(=O)[C@@H]3CCCN3C(=O)c3ccno3)cc2)cc1)[C@@H]1CCCN1C(=O)c1ccno1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
RHOC P08134 1/20 0.46
RHOA P61586 1/20 0.46
ALDH1A1 P00352 2/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
MAPT P10636 1/20 0.42
HTT P42858 2/20 0.42
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
NPC1 O15118 1/20 0.41
TRPV1 Q8NER1 1/20 0.41
MAPK1 P28482 1/20 0.41
HSD17B10 Q99714 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL845182 0.81 HSD17B10 (0.57) RHOCRHOAALDH1A1CYP2C9CYP2C19
SCHEMBL844934 0.81 RHOC (0.51) RHOCRHOAALDH1A1CYP2C9CYP2C19
SCHEMBL873200 0.79 RHOC (0.48) RHOCRHOAALDH1A1CYP2C9CYP2C19
SCHEMBL845403 0.79 GFER (0.46) RHOCRHOAALDH1A1CYP2C9CYP2C19
SCHEMBL845300 0.78 CYP2C9 (0.54) RHOCRHOAALDH1A1CYP2C9CYP2C19
SCHEMBL845405 0.78 TRPV1 (0.46) RHOCRHOACYP2C9CYP2C19MAPT
SCHEMBL845048 0.78 DGAT1 (0.50) RHOCRHOAALDH1A1CYP2C9CYP2C19
SCHEMBL845297 0.77 RHOC (0.48) RHOCRHOAALDH1A1CYP2C9CYP2C19
SCHEMBL4887329 0.77 CA2 (0.48) ALDH1A1KMT2A
SCHEMBL4887332 0.77 CA2 (0.48) ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed