SCHEMBL845313

SCHEMBL845313

Cc1cccc(C(=O)N2CCC[C@H]2C(=O)Nc2ccc(/C=C/c3ccc(NC(=O)[C@@H]4CCCN4)cc3)cc2)n1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.41
SCN9A Q15858 2/20 0.41
POLB P06746 1/20 0.41
SCN3A Q9NY46 1/20 0.41
SCN5A Q14524 1/20 0.41
DHODH Q02127 2/20 0.40
SIRT2 Q8IXJ6 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
KHK P50053 2/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
DGAT1 O75907 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL845367 0.91 ALDH1A1 (0.47) ALDH1A1POLBCYP2C9CYP2C19MEN1
SCHEMBL10119551 0.82 DHODH (0.40) ALDH1A1SCN9APOLBSCN3ASCN5A
SCHEMBL872532 0.82 TRPV1 (0.44) ALDH1A1CYP2C9CYP2C19
SCHEMBL873223 0.81 RHOC (0.43) SCN9ASCN3ASCN5AMEN1KMT2A
SCHEMBL872886 0.80 KDM4E (0.52) ALDH1A1POLBMEN1KMT2A
SCHEMBL874324 0.80 MAPK1 (0.42) ALDH1A1CYP2C9CYP2C19
SCHEMBL10119294 0.80 ITGB3 (0.41) ALDH1A1SCN9ASCN3A
SCHEMBL874056 0.80 TRPV1 (0.42) ALDH1A1CYP2C9CYP2C19MEN1KMT2A
SCHEMBL871556 0.80 CYP2C9 (0.38) ALDH1A1SCN9ASCN3ASCN5ACYP2C9
SCHEMBL874313 0.79 MAPK1 (0.50) ALDH1A1CYP2C9CYP2C19MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed