SCHEMBL847277

SCHEMBL847277

O=Cc1ccc(S(=O)(=O)N2CCOCC2)cc1

nearest known ligand 0.69

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
POLB P06746 3/20 0.69
LMNA P02545 4/20 0.63
SMN1; SMN2 Q16637 3/20 0.63
KMT2A Q03164 2/20 0.61
GAA P10253 2/20 0.61
MEN1 O00255 1/20 0.61
L3MBTL1 Q9Y468 2/20 0.56
MAPK1 P28482 1/20 0.56
ALDH1A1 P00352 3/20 0.55
KDM4E B2RXH2 2/20 0.55
HSD17B10 Q99714 2/20 0.55
TSHR P16473 2/20 0.55
USP2 O75604 1/20 0.55
HTT P42858 1/20 0.55
APOBEC3G Q9HC16 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12793245 0.87 POLB (0.88) POLBLMNASMN1; SMN2KMT2AGAA
SCHEMBL29687970 0.85 POLB (0.67) POLBLMNASMN1; SMN2KMT2AGAA
SCHEMBL1987080 0.84 USP2 (0.70) POLBLMNASMN1; SMN2KMT2AGAA
SCHEMBL5804200 0.82 USP2 (0.74) POLBLMNASMN1; SMN2KMT2AGAA
SCHEMBL2798288 0.82 USP2 (0.74) POLBLMNASMN1; SMN2KMT2AGAA
SCHEMBL4811982 0.82 POLB (0.63) POLBLMNASMN1; SMN2KMT2AGAA
SCHEMBL7267448 0.82 POLB (0.63) POLBLMNASMN1; SMN2KMT2AGAA
SCHEMBL3591766 0.82 POLB (0.63) POLBLMNASMN1; SMN2KMT2AGAA
SCHEMBL12793258 0.82 POLB (1.00) POLBLMNASMN1; SMN2KMT2AGAA
SCHEMBL12793309 0.81 POLB (0.67) POLBLMNASMN1; SMN2KMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 34 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230142739-A1 PROTEIN-PROTEIN INTERACTION STABILIZERS UNIV CALIFORNIA (US) 2023-05-11 US disclosed
EP-4125861-A2 PROTEIN-PROTEIN INTERACTION STABILIZERS The Regents of the University of California (US) 2023-02-08 EP disclosed
CN-105008350-B Antiviral compound 弗·哈夫曼-拉罗切有限公司 2018-05-08 CN disclosed
EP-2964637-B1 ANTIVIRAL COMPOUNDS HOFFMANN LA ROCHE (CH) 2017-04-12 EP disclosed
US-9428469-B2 Antiviral compounds HOFFMANN-LA ROCHE (US) 2016-08-30 US disclosed
US-20160009666-A1 ANTIVIRAL COMPOUNDS HOFFMANN-LA ROCHE INC. 2016-01-14 US disclosed
EP-2964637-A1 ANTIVIRAL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2016-01-13 EP disclosed
CN-105008350-A Antiviral compounds HOFFMANN LA ROCHE HOFFMANN LA ROCHE 2015-10-28 CN disclosed
WO-2014135422-A1 ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2014-09-12 WO disclosed
US-8163906-B2 Dihydroquinone and dihydronaphthridine inhibitors of JNK ROCHE PALO ALTO, LLC (US) 2012-04-24 US disclosed
EP-1753714-A4 2-SUBSTITUTED AND 4-SUBSTITUTED ARYL NITRONE COMPOUDS RENOVIS INC (US) 2007-10-17 EP disclosed
EP-1753714-A2 2-SUBSTITUTED AND 4-SUBSTITUTED ARYL NITRONE COMPOUDS Renovis, Inc. (US) 2007-02-21 EP disclosed
US-20060264460-A1 3-Cyanoquinoline inhibitors of Tpl2 kinase and methods of making and using the same WYETH (US) 2006-11-23 US disclosed
WO-2006124692-A2 3-CYANOQUINOLINE INHIBITORS OF TPL2 KINASE AND METHODS OF MAKING AND USING THE SAME WYETH (US) 2006-11-23 WO disclosed
WO-2006093518-A2 THIENYL COMPOUNDS FOR TREATING VIRUS-RELATED CONDITIONS APATH, LLC (US) 2006-09-08 WO disclosed
US-20050256159-A1 1,4-disubstituted piperidine derivatives and their use as 11,betahsd1 inhibitors ASTRAZENECA AB (SE) 2005-11-17 US disclosed
WO-2005079270-A2 2-SUBSTITUTED AND 4-SUBSTITUTED ARYL NITRONE COMPOUDS RENOVIS, INC. (US) 2005-09-01 WO disclosed
US-20050182060-A1 2-Substituted and 4-substituted aryl nitrone compounds RENOVIS, INC. 2005-08-18 US disclosed
EP-1556349-A1 1,4-DISUBSTITUTED PIPERIDINE DERIVATIVES AND THEIR USE AS 11-BETAHSD1 INHIBITORS Astrazeneca AB (SE) 2005-07-27 EP disclosed
WO-2004033427-A1 1,4-DISUBSTITUTED PIPERIDINE DERIVATIVES AND THEIR USE AS 11-BETAHSD1 INHIBITORS ASTRAZENECA AB (SE) 2004-04-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160009666-A1 ANTIVIRAL COMPOUNDS HAVCR2, EIF2AK2, MAVS POLB 863/4885LMNA 3788/4885SMN1; SMN2 2807/4885
US-20050182060-A1 2-Substituted and 4-substituted aryl nitrone compounds CXCR2, CCL5, CCL2 POLB 1976/4885LMNA 3216/4885SMN1; SMN2 1311/4885
US-20230142739-A1 PROTEIN-PROTEIN INTERACTION STABILIZERS HSPBP1, HSPA8, HSPH1 POLB 3568/4885LMNA 2827/4885SMN1; SMN2 1672/4885
US-20050256159-A1 1,4-disubstituted piperidine derivatives and their use as 11,betahsd1 inhibitors HSD11B1, HSD3B1, P4HA1 POLB 1926/4885LMNA 3152/4885SMN1; SMN2 3573/4885
US-20060264460-A1 3-Cyanoquinoline inhibitors of Tpl2 kinase and methods of making and using the same TNNI3K, CSNK1A1L, CDKL1 POLB 2825/4885LMNA 2364/4885SMN1; SMN2 4362/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.