SCHEMBL8494571

SCHEMBL8494571

Cc1ccc(S(=O)(=O)NCCCNCCCCNCCCN)cc1

nearest known ligand 0.65

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 14/20 0.65
CA12 O43570 1/20 0.57
CA2 P00918 1/20 0.57
CA9 Q16790 1/20 0.57
ALOX15 P16050 1/20 0.56
MEN1 O00255 2/20 0.54
KMT2A Q03164 2/20 0.54
HTT P42858 2/20 0.53
MBTD1 Q05BQ5 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
LMNA P02545 3/20 0.52
NPSR1 Q6W5P4 1/20 0.52
GAA P10253 1/20 0.51
MAPT P10636 1/20 0.51
PKM P14618 1/20 0.50
HPGD P15428 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13426054 0.95 ALDH1A1 (0.62) ALDH1A1CA12CA2CA9ALOX15
SCHEMBL7628596 0.92 ALDH1A1 (0.70) ALDH1A1CA12CA2CA9ALOX15
SCHEMBL7955008 0.91 ALDH1A1 (0.68) ALDH1A1CA12CA2CA9ALOX15
SCHEMBL3969095 0.91 ALDH1A1 (0.72) ALDH1A1CA12CA2CA9ALOX15
SCHEMBL17599857 0.89 ALDH1A1 (0.66) ALDH1A1CA12CA2CA9ALOX15
SCHEMBL12849347 0.89 ALDH1A1 (0.66) ALDH1A1CA12CA2CA9ALOX15
Hydrochloric Acid SCHEMBL11629317 0.88 ALDH1A1 (0.64) ALDH1A1CA12CA2CA9ALOX15
Hydrochloric Acid SCHEMBL5093423 0.88 ALDH1A1 (0.64) ALDH1A1CA12CA2CA9ALOX15
SCHEMBL12085676 0.87 ALDH1A1 (0.67) ALDH1A1HTTL3MBTL1LMNANPSR1
SCHEMBL7937849 0.86 ALDH1A1 (0.62) ALDH1A1CA12CA2CA9ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10350178-B2 Methods and compositions for treatment of demyelinating diseases PATHOLOGICA LLC (US) 2019-07-16 US disclosed
US-20170290788-A1 PHARMACEUTICAL FOR ORAL DELIVERY COMPRISING MGBG AND METHODS OF TREATING DISEASE PATHOLOGICA, LLC 2017-10-12 US disclosed
US-9616035-B2 Pharmaceutical for oral delivery comprising MGBG and methods of treating disease PATHOLOGICA, LLC (US) 2017-04-11 US disclosed
US-20150359761-A1 METHODS AND COMPOSITIONS FOR TREATMENT OF DEMYELINATING DISEASES PATHOLOGICA, LLC 2015-12-17 US disclosed
WO-2014110154-A1 METHODS AND COMP0STIONS FOR TREATMENT OF DEMYELINATING DISEASES PATHOLOGICA LLC (US) 2014-07-17 WO disclosed
US-8779195-B2 Polyamine derivatives NIHON UNIVERSITY (JP) 2014-07-15 US disclosed
US-8779195-B2 Polyamine derivatives NIHON UNIVERSITY (JP) 2014-07-15 US disclosed
US-20140051765-A1 PHARMACEUTICAL FOR ORAL DELIVERY COMPRISING MGBG AND METHODS OF TREATING DISEASE PATHOLOGICA LLC (US) 2014-02-20 US disclosed
US-20120289604-A1 PHARMACEUTICAL FOR ORAL DELIVERY COMPRISING MGBG AND METHODS OF TREATING DISEASE PATHOLOGICA LLC (US) 2012-11-15 US disclosed
US-8258186-B2 Pharmaceutical for oral delivery comprising MGBG PATHOLOGICA, LLC (US) 2012-09-04 US disclosed
US-20110112199-A1 PHARMACEUTICAL FOR ORAL DELIVERY COMPRISING MGBG AND METHODS OF TREATING DISEASE PATHOLOGICA LLC (US) 2011-05-12 US disclosed
WO-2011009039-A2 PHARMACEUTICAL FOR ORAL DELIVERY COMPRISING MGBG AND METHODS OF TREATING DISEASE PATHOLOGICA LLC (US) 2011-01-20 WO disclosed
US-20100063322-A1 NOVEL POLYAMINE DERIVATIVES NIHON UNIVERSITY (JP) 2010-03-11 US disclosed
US-5866613-A Anti-neoplastic, anti-viral or anti-retroviral spermine derivatives UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 1999-02-02 US disclosed
US-5342945-A Bis-hexahydropyrimidinylakyl compounds UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 1994-08-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100063322-A1 NOVEL POLYAMINE DERIVATIVES SRM, SMS, H1-3 ALDH1A1 3019/4885CA12 2932/4885CA2 1327/4885
US-20150359761-A1 METHODS AND COMPOSITIONS FOR TREATMENT OF DEMYELINATING DISEASES SRM, PMP22, SMS ALDH1A1 2747/4885CA12 4738/4885CA2 4344/4885
US-20140051765-A1 PHARMACEUTICAL FOR ORAL DELIVERY COMPRISING MGBG AND METHODS OF TREATING DISEASE BPGM, PYGB, EDNRB ALDH1A1 1462/4885CA12 2977/4885CA2 3322/4885
US-20170290788-A1 PHARMACEUTICAL FOR ORAL DELIVERY COMPRISING MGBG AND METHODS OF TREATING DISEASE BPGM, PYGB, EDNRB ALDH1A1 1462/4885CA12 2977/4885CA2 3322/4885
US-20120289604-A1 PHARMACEUTICAL FOR ORAL DELIVERY COMPRISING MGBG AND METHODS OF TREATING DISEASE BPGM, PYGB, EDNRB ALDH1A1 1462/4885CA12 2977/4885CA2 3322/4885
US-20110112199-A1 PHARMACEUTICAL FOR ORAL DELIVERY COMPRISING MGBG AND METHODS OF TREATING DISEASE BPGM, PYGB, EDNRB ALDH1A1 1462/4885CA12 2977/4885CA2 3322/4885
US-10350178-B2 Methods and compositions for treatment of demyelinating diseases PMP22, MAG, GMFG ALDH1A1 2637/4885CA12 1122/4885CA2 2259/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.