SCHEMBL8495236

SCHEMBL8495236

CCCCCN1c2ccccc2C=CC1C#N

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.42
LMNA P02545 5/20 0.42
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
MAPT P10636 4/20 0.36
SMN1; SMN2 Q16637 3/20 0.36
THRB P10828 2/20 0.36
MAPK1 P28482 1/20 0.36
HTT P42858 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
ALDH2 P05091 1/20 0.35
ALDH3A1 P30838 1/20 0.35
CES1 P23141 2/20 0.34
CDC25A P30304 2/20 0.34
KDM4E B2RXH2 2/20 0.33
GLA P06280 1/20 0.33
POLB P06746 1/20 0.33
GAA P10253 1/20 0.33
HPGD P15428 1/20 0.33
CASP1 P29466 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28295668 0.78 LMNA (0.41) ALDH1A1LMNAMEN1KMT2ASMN1; SMN2
SCHEMBL28486552 0.74 PRKCG (0.37) ALDH1A1LMNAMEN1KMT2AMAPT
SCHEMBL10613637 0.69 PTGS1 (0.53) ALDH1A1MEN1KMT2AMAPTMAPK1
SCHEMBL5323524 0.67 CES1 (0.53) ALDH1A1MEN1KMT2AMAPTMAPK1
SCHEMBL28537893 0.67 CES1 (0.45) ALDH1A1LMNAMEN1KMT2AALDH2
SCHEMBL32677342 0.67 NR1H2 (0.38) ALDH1A1LMNASMN1; SMN2MAPK1ALDH2
SCHEMBL11036624 0.67 ATM (0.46) ALDH1A1LMNAMEN1KMT2AMAPT
Bromide SCHEMBL460851 0.64 ALDH1A1 (0.47) ALDH1A1LMNAMEN1KMT2AMAPT
SCHEMBL4595897 0.64 KMT2A (0.47) ALDH1A1LMNAMEN1KMT2AMAPT
SCHEMBL28461113 0.63 TDP1 (0.39) ALDH1A1LMNAMEN1KMT2ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5939435-A TREATMENT OF ATHEROSCLEROSIS AND CORONARY HEART DISEASE AMERICAN HOME PRODUCTS CORPORATION (US) 1999-08-17 US disclosed
US-4194987-A N-ACYL-CYANO-DIHYDRO(ISO)QUINOLINES AS ACTIVATORS FMC CORPORATION (US) 1980-03-25 US disclosed