SCHEMBL8515925

SCHEMBL8515925

CCOC(=O)c1c(-c2ccc(-c3ccc(Cl)cc3)cc2)[nH]c2ccccc2c1=O

nearest known ligand 0.64

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 7/20 0.64
PTGES O14684 4/20 0.64
MEN1 O00255 2/20 0.60
LMNA P02545 2/20 0.60
MAPT P10636 2/20 0.60
KMT2A Q03164 2/20 0.60
TP53 P04637 1/20 0.55
MDM2 Q00987 1/20 0.55
CSF1R P07333 1/20 0.55
KDM4E B2RXH2 2/20 0.54
ALDH1A1 P00352 2/20 0.54
HPGD P15428 2/20 0.54
GAA P10253 1/20 0.54
MAPK10 P53779 1/20 0.54
HSD17B10 Q99714 1/20 0.54
NPC1 O15118 1/20 0.51
CYP1A2 P05177 1/20 0.49
XBP1 P17861 1/20 0.49
CYP2C19 P33261 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6300719 0.89 ALDH1A1 (0.67) ALOX5MEN1LMNAMAPTKMT2A
SCHEMBL8512850 0.88 MEN1 (0.56) ALOX5PTGESMEN1LMNAMAPT
SCHEMBL6295725 0.86 CSF1R (0.71) ALOX5PTGESMEN1LMNAMAPT
SCHEMBL8512448 0.84 KMT2A (0.50) ALOX5PTGESMEN1LMNAMAPT
SCHEMBL6300423 0.83 ALOX5 (0.55) ALOX5PTGESMEN1LMNAMAPT
SCHEMBL3555503 0.82 AR (0.58) MEN1LMNAMAPTKMT2AKDM4E
SCHEMBL19846945 0.80 KDM4E (0.58) ALOX5MEN1LMNAMAPTKMT2A
SCHEMBL30482846 0.79 ALDH1A1 (0.76) ALOX5PTGESMEN1LMNAMAPT
SCHEMBL6300618 0.78 ALOX5 (0.60) ALOX5PTGESMEN1LMNAMAPT
SCHEMBL8512623 0.78 NPC1 (0.47) ALOX5PTGESMEN1LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10799494-B2 Combination of respiratory electron transport chain inhibitors with a cytochrome bd inhibitor LIVERPOOL SCHOOL TROPICAL MEDICINE (GB) 2020-10-13 US claimed
US-20190151305-A1 COMBINATION PRODUCT LIVERPOOL SCHOOL TROPICAL MEDICINE (GB) 2019-05-23 US claimed
EP-3389659-A1 COMBINATION PRODUCT Liverpool School of Tropical Medicine (GB) 2018-10-24 EP claimed
WO-2017103615-A1 COMBINATION PRODUCT LIVERPOOL SCHOOL OF TROPICAL MEDICINE (GB) 2017-06-22 WO claimed
WO-2012069856-A1 ANTIMALARIAL COMPOUNDS LIVERPOOL SCHOOL OF TROPICAL MEDICINE (GB) 2012-05-31 WO claimed
US-10799494-B2 Combination of respiratory electron transport chain inhibitors with a cytochrome bd inhibitor LIVERPOOL SCHOOL TROPICAL MEDICINE (GB) 2020-10-13 US disclosed
US-10799494-B2 Combination of respiratory electron transport chain inhibitors with a cytochrome bd inhibitor LIVERPOOL SCHOOL TROPICAL MEDICINE (GB) 2020-10-13 US disclosed
US-20190151305-A1 COMBINATION PRODUCT LIVERPOOL SCHOOL TROPICAL MEDICINE (GB) 2019-05-23 US disclosed
US-20190151305-A1 COMBINATION PRODUCT LIVERPOOL SCHOOL TROPICAL MEDICINE (GB) 2019-05-23 US disclosed
EP-3389659-A1 COMBINATION PRODUCT Liverpool School of Tropical Medicine (GB) 2018-10-24 EP disclosed
WO-2017103615-A1 COMBINATION PRODUCT LIVERPOOL SCHOOL OF TROPICAL MEDICINE (GB) 2017-06-22 WO disclosed
WO-2017103615-A1 COMBINATION PRODUCT LIVERPOOL SCHOOL OF TROPICAL MEDICINE (GB) 2017-06-22 WO disclosed
WO-2012069856-A1 ANTIMALARIAL COMPOUNDS LIVERPOOL SCHOOL OF TROPICAL MEDICINE (GB) 2012-05-31 WO disclosed
WO-2012069856-A1 ANTIMALARIAL COMPOUNDS LIVERPOOL SCHOOL OF TROPICAL MEDICINE (GB) 2012-05-31 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10799494-B2 Combination of respiratory electron transport chain inhibitors with a cytochrome bd inhibitor NDUFB7, NDUFB3, NDUFB5 ALOX5 3066/4885PTGES 967/4885MEN1 4848/4885
US-20190151305-A1 COMBINATION PRODUCT NDUFB5, NDUFB7, NDUFB10 ALOX5 2373/4885PTGES 823/4885MEN1 4581/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.