SCHEMBL8519376

SCHEMBL8519376

CC(C)(C)OC(=O)NCc1cccc(C2(CC(=O)O)CN(CCc3ccccc3)C(=O)c3ccccc3N2C(N)=O)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 1/20 0.39
PDCD1 Q15116 1/20 0.38
CD274 Q9NZQ7 1/20 0.38
BRD4 O60885 1/20 0.38
CREBBP Q92793 1/20 0.38
SIGMAR1 Q99720 3/20 0.35
GLS O94925 2/20 0.34
UTS2R Q9UKP6 3/20 0.34
ALDH1A1 P00352 1/20 0.34
TSHR P16473 1/20 0.34
BRD9 Q9H8M2 1/20 0.34
BAZ2B Q9UIF8 1/20 0.34
BAZ2A Q9UIF9 1/20 0.34
NPC1 O15118 1/20 0.34
TP53 P04637 1/20 0.34
POLB P06746 1/20 0.34
RAB9A P51151 1/20 0.34
AKT1 P31749 1/20 0.33
NSD2 O96028 1/20 0.33
DRD2 P14416 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8518279 0.92 AKT1 (0.37) CCKBRPDCD1CD274BRD4CREBBP
SCHEMBL8518520 0.82 MAPT (0.39) ALDH1A1NPC1TP53RAB9A
SCHEMBL8518880 0.73 NAMPT (0.45) CCKBRSIGMAR1ALDH1A1AKT1DRD2
SCHEMBL7400533 0.71 CCKBR (0.49) CCKBRPDCD1CD274BRD4CREBBP
SCHEMBL7394047 0.67 NAMPT (0.49) CCKBRPDCD1CD274DRD2NAMPT
SCHEMBL21996778 0.65 POLB (0.51) PDCD1CD274ALDH1A1TSHRBRD9
SCHEMBL31608963 0.64 KMT2A (0.51) CCKBRPDCD1CD274BRD4CREBBP
SCHEMBL3838871 0.62 CA12 (0.63) ALDH1A1RAB9AAKT1NAMPT
SCHEMBL5729298 0.62 GLS (0.54) BRD4CREBBPGLS
SCHEMBL29072723 0.62 BRD4 (0.48) CCKBRBRD4CREBBPGLSBRD9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5939412-A Bicyclic fibrinogen antagonists SMITHKLINE BEECHAM CORPORATION (US) 1999-08-17 US disclosed
US-5693636-A Bicyclic fibrinogen antagonists SMITHKLINE BEECHAM CORPORATION (US) 1997-12-02 US disclosed