SCHEMBL8518880

SCHEMBL8518880

CC(C)(C)OC(=O)NCc1ccc(C2(CC(=O)O)C(=O)N(CCc3ccccc3)Cc3ccccc3N2C(N)=O)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 2/20 0.45
DRD2 P14416 2/20 0.39
CACNA1G O43497 3/20 0.37
CACNA1H O95180 3/20 0.37
CACNA1I Q9P0X4 3/20 0.37
SIGMAR1 Q99720 3/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
PARP1 P09874 1/20 0.35
PARP2 Q9UGN5 1/20 0.35
MTNR1A P48039 1/20 0.35
MTNR1B P49286 1/20 0.35
HDAC1 Q13547 1/20 0.35
AKT1 P31749 1/20 0.34
SCN9A Q15858 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPK10 P53779 1/20 0.33
CCKBR P32239 1/20 0.33
PSMB1 P20618 1/20 0.33
PSMB8 P28062 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8401265 0.81 ITGB3 (0.44) PARP1PARP2
SCHEMBL8897079 0.80 PARP1 (0.39) CACNA1GCACNA1HCACNA1IPARP1PARP2
SCHEMBL8518279 0.79 AKT1 (0.37) NAMPTDRD2SIGMAR1MEN1KMT2A
SCHEMBL7400352 0.73 NAMPT (0.55) NAMPTDRD2CACNA1GCACNA1HCACNA1I
SCHEMBL8519376 0.73 CCKBR (0.39) NAMPTDRD2SIGMAR1AKT1ALDH1A1
SCHEMBL7437642 0.67 ITGB3 (0.65)
SCHEMBL7437648 0.67 ITGB3 (0.65)
SCHEMBL3838871 0.66 CA12 (0.63) NAMPTMEN1KMT2AHDAC1AKT1
SCHEMBL7394047 0.66 NAMPT (0.49) NAMPTDRD2CACNA1GCACNA1HCACNA1I
SCHEMBL7241814 0.65 HDAC1 (0.44) NAMPTCACNA1GSIGMAR1HDAC1AKT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5939412-A Bicyclic fibrinogen antagonists SMITHKLINE BEECHAM CORPORATION (US) 1999-08-17 US disclosed
US-5693636-A Bicyclic fibrinogen antagonists SMITHKLINE BEECHAM CORPORATION (US) 1997-12-02 US disclosed