SCHEMBL8520753

SCHEMBL8520753

CC/C(=C\c1ccc(NC(=O)c2cccc(NC(=N)N)c2)cc1)C(=O)O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.48
MEN1 O00255 2/20 0.48
NPC1 O15118 1/20 0.48
POLB P06746 1/20 0.47
ITGB3 P05106 3/20 0.45
ITGA2B P08514 3/20 0.45
KCNK3 O14649 1/20 0.45
KCNK9 Q9NPC2 1/20 0.45
NR1H4 Q96RI1 2/20 0.43
PLK4 O00444 1/20 0.43
CHEK1 O14757 1/20 0.43
AURKA O14965 1/20 0.43
CHUK O15111 1/20 0.43
DAPK3 O43293 1/20 0.43
JAK2 O60674 1/20 0.43
ROCK2 O75116 1/20 0.43
PAK4 O96013 1/20 0.43
CHEK2 O96017 1/20 0.43
CDK1 P06493 1/20 0.43
PIM1 P11309 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8520762 0.85 KMT2A (0.44) KMT2AMEN1NPC1POLBITGB3
SCHEMBL8520922 0.84 FFAR1 (0.46) KMT2AMEN1NPC1ITGB3ITGA2B
SCHEMBL7572346 0.84 ITGB3 (0.50) KMT2AMEN1NPC1POLBITGB3
SCHEMBL7498232 0.83 NR1H4 (0.41) KMT2AMEN1NPC1POLBITGB3
SCHEMBL7506955 0.80 KMT2A (0.50) KMT2AMEN1NPC1POLBKCNK3
SCHEMBL7497380 0.80 KMT2A (0.50) KMT2AMEN1NPC1POLBKCNK3
SCHEMBL8538573 0.80 EPHX2 (0.41) KMT2AMEN1POLBKCNK3KCNK9
SCHEMBL8520757 0.79 KMT2A (0.51) KMT2AMEN1NPC1POLBITGB3
SCHEMBL7506884 0.78 ITGB3 (0.66) KMT2ANPC1POLBITGB3ITGA2B
SCHEMBL7508818 0.78 ITGB3 (0.66) KMT2ANPC1POLBITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0894084-A1 CINNAMIC ACID DERIVATIVES AND THEIR USE AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1999-02-03 EP disclosed
WO-1997036860-A1 CINNAMIC ACID DERIVATIVES AND THEIR USE AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1997-10-09 WO disclosed