SCHEMBL8526941

SCHEMBL8526941

CCC(CC)C(=O)NOC(=O)CC(=O)OCc1ccc(N)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPID Q08752 2/20 0.39
PPIB P23284 1/20 0.39
PPIA P62937 1/20 0.39
PPIG Q13427 1/20 0.39
CA1 P00915 4/20 0.37
CA2 P00918 3/20 0.37
CA7 P43166 2/20 0.37
CA14 Q9ULX7 2/20 0.37
ALDH1A1 P00352 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
CYP1A2 P05177 3/20 0.36
CYP3A4 P08684 3/20 0.36
CYP2C9 P11712 2/20 0.36
CYP2C19 P33261 2/20 0.36
CYP2D6 P10635 1/20 0.36
ABCC3 O15438 1/20 0.36
NR1I2 O75469 1/20 0.36
ABCB11 O95342 1/20 0.36
NR3C1 P04150 1/20 0.36
RARG P13631 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8528385 0.85 THRA (0.36) ALDH1A1SMN1; SMN2CYP1A2CYP3A4CYP2C9
SCHEMBL8422211 0.83 ALDH1A1 (0.38) CA1CA2CA7CA14ALDH1A1
SCHEMBL2781111 0.81 PPIB (0.40) PPIDPPIBPPIAPPIGCA1
SCHEMBL6453211 0.81 ALDH1A1 (0.47) PPIDPPIBPPIAPPIGCA1
SCHEMBL19439087 0.79 PPID (0.57) PPIDPPIBPPIAPPIGALDH1A1
SCHEMBL1428501 0.77 TSHR (0.48) CA1CA2CA7CA14ALDH1A1
SCHEMBL23623825 0.75 PPID (0.46) PPIDPPIBPPIAPPIGCA1
SCHEMBL11736357 0.75 PPIB (0.44) PPIDPPIBPPIAPPIGCA1
SCHEMBL8422387 0.74 CTSL (0.35) ALDH1A1SMN1; SMN2LMNA
SCHEMBL10082417 0.74 CYP1A2 (0.47) PPIDPPIBPPIAPPIGCA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0705257-B1 AMINOACID DERIVATIVES AS NO SYNTHASE INHIBITORS WELLCOME FOUND (GB) 1998-03-11 EP disclosed
EP-0705257-A1 AMINOACID DERIVATIVES AS NO SYNTHASE INHIBITORS THE WELLCOME FOUNDATION LIMITED (GB) 1996-04-10 EP disclosed
WO-1995000505-A1 AMINOACID DERIVATIVES AS NO SYNTHASE INHIBITORS THE WELLCOME FOUNDATION LIMITED (GB) 1995-01-05 WO disclosed