SCHEMBL8528385

SCHEMBL8528385

CCC(CC)C(=O)NOC(=O)CC(=O)OCc1cccc(N)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRA P10827 1/20 0.36
THRB P10828 1/20 0.36
POLB P06746 1/20 0.35
PKM P14618 1/20 0.34
KMT2A Q03164 1/20 0.34
TACR1 P25103 1/20 0.34
HTT P42858 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
ALDH1A1 P00352 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
SLC7A5 Q01650 1/20 0.34
GLA P06280 1/20 0.34
SLC15A1 P46059 1/20 0.34
KDM4E B2RXH2 1/20 0.34
MAPT P10636 1/20 0.34
RAB9A P51151 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8526941 0.85 PPID (0.39) HTTNPSR1ALDH1A1SMN1; SMN2MAPT
SCHEMBL2780510 0.83 ALDH1A1 (0.42) THRATHRBPOLBTACR1ALDH1A1
SCHEMBL8422387 0.82 CTSL (0.35) KMT2ATACR1ALDH1A1SMN1; SMN2LMNA
SCHEMBL14416816 0.77 THRA (0.44) THRATHRBNPSR1ALDH1A1SMN1; SMN2
SCHEMBL3911621 0.74 ALDH1A1 (0.45) THRATHRBPOLBTACR1ALDH1A1
SCHEMBL8422211 0.74 ALDH1A1 (0.38) KMT2ATACR1ALDH1A1SMN1; SMN2MAPT
SCHEMBL27615700 0.73 SLC15A1 (0.45) THRATHRBPOLBTACR1ALDH1A1
SCHEMBL1428501 0.73 TSHR (0.48) KMT2AHTTNPSR1ALDH1A1SMN1; SMN2
SCHEMBL21385079 0.72 THRA (0.45) THRATHRBALDH1A1GLAKDM4E
SCHEMBL11830714 0.72 FOLH1 (0.48) KMT2ASMN1; SMN2SLC7A5PPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0705257-B1 AMINOACID DERIVATIVES AS NO SYNTHASE INHIBITORS WELLCOME FOUND (GB) 1998-03-11 EP disclosed
EP-0705257-A1 AMINOACID DERIVATIVES AS NO SYNTHASE INHIBITORS THE WELLCOME FOUNDATION LIMITED (GB) 1996-04-10 EP disclosed
WO-1995000505-A1 AMINOACID DERIVATIVES AS NO SYNTHASE INHIBITORS THE WELLCOME FOUNDATION LIMITED (GB) 1995-01-05 WO disclosed