SCHEMBL8422211

SCHEMBL8422211

CCC(CC)C(=O)NOC(=O)CC(=O)OCc1ccc(NC#N)cc1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
RAB9A P51151 1/20 0.36
CTSL P07711 10/20 0.35
CTSS P25774 10/20 0.35
CTSB P07858 8/20 0.35
CTSK P43235 6/20 0.35
CA1 P00915 3/20 0.34
CA2 P00918 3/20 0.34
CA7 P43166 2/20 0.34
CA14 Q9ULX7 2/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
TACR1 P25103 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8422387 0.87 CTSL (0.35) ALDH1A1SMN1; SMN2CTSLCTSSCTSB
SCHEMBL8526941 0.83 PPID (0.39) ALDH1A1SMN1; SMN2RAB9ACA1CA2
SCHEMBL8528385 0.74 THRA (0.36) ALDH1A1SMN1; SMN2RAB9AKMT2ATACR1
SCHEMBL1428501 0.71 TSHR (0.48) ALDH1A1SMN1; SMN2RAB9ACA1CA2
SCHEMBL27611926 0.69 TSHR (0.43) ALDH1A1SMN1; SMN2RAB9A
SCHEMBL21652695 0.65 MGAM (0.62) ALDH1A1MEN1KMT2AMAPT
SCHEMBL8978333 0.65 ALDH1A1 (0.44) ALDH1A1SMN1; SMN2CTSLCTSSCTSB
SCHEMBL27630941 0.65 TPSAB1 (0.44) ALDH1A1SMN1; SMN2CA1CA2MEN1
SCHEMBL27611924 0.65 KDM4E (0.39) ALDH1A1SMN1; SMN2CA1CA2MEN1
SCHEMBL2781111 0.65 PPIB (0.40) ALDH1A1SMN1; SMN2CA1CA2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5874472-A Aminoacid derivatives as no synthase inhibitors GLAXO WELLCOME INC. (US) 1999-02-23 US disclosed
EP-0705257-B1 AMINOACID DERIVATIVES AS NO SYNTHASE INHIBITORS WELLCOME FOUND (GB) 1998-03-11 EP disclosed
EP-0705257-A1 AMINOACID DERIVATIVES AS NO SYNTHASE INHIBITORS THE WELLCOME FOUNDATION LIMITED (GB) 1996-04-10 EP disclosed
WO-1995000505-A1 AMINOACID DERIVATIVES AS NO SYNTHASE INHIBITORS THE WELLCOME FOUNDATION LIMITED (GB) 1995-01-05 WO disclosed