SCHEMBL8529307

SCHEMBL8529307

COc1cc(CSc2ccc(O)cc2)cc(OC)c1OC

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.50
CYP3A4 P08684 1/20 0.48
MAPT P10636 1/20 0.48
TUBB4A P04350 7/20 0.48
TUBB P07437 7/20 0.48
TUBA3C P0DPH7 7/20 0.48
TUBA1B P68363 7/20 0.48
TUBA4A P68366 7/20 0.48
TUBB4B P68371 7/20 0.48
TUBB3 Q13509 7/20 0.48
TUBB2A Q13885 7/20 0.48
TUBB8 Q3ZCM7 7/20 0.48
TUBA3E Q6PEY2 7/20 0.48
TUBA1A Q71U36 7/20 0.48
TUBA1C Q9BQE3 7/20 0.48
TUBB6 Q9BUF5 7/20 0.48
TUBB2B Q9BVA1 7/20 0.48
TUBB1 Q9H4B7 7/20 0.48
BACE1 P56817 1/20 0.43
GALR3 O60755 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8530817 0.89 EGFR (0.46) MAPTALDH1A1
SCHEMBL8529682 0.86 AKR1B1 (0.46) CYP3A4TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL6338880 0.85 TUBB4A (0.60) PTGS2TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL8530355 0.83 CA2 (0.48) PTGS2TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL9089503 0.76 TUBB4A (0.71) PTGS2CYP3A4MAPTTUBB4ATUBB
SCHEMBL4542980 0.75 LTA4H (0.50) CYP3A4ALDH1A1TSHRRAB9ACA9
SCHEMBL9475495 0.75 APP (0.70) MAPTRAB9ASMN1; SMN2
SCHEMBL10126440 0.74 ABL1 (0.43) PTGS2CYP3A4MAPTRAB9ASMN1; SMN2
SCHEMBL14139160 0.74 TUBB4A (0.40) PTGS2TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL10614759 0.73 PTGS2 (0.61) PTGS2CYP3A4MAPTTUBB4ATUBB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5840991-A 3,4,5-TRIHYDROXYBENZYL-4-HYDROXYPHENYL THIOETHER DEVELOPMENT CENTER FOR BIOTECHNOLOGY (TW) 1998-11-24 US claimed
US-7410998-B2 Inhibitors of NADH:ubiquinone oxidoreductase THE SCRIPPS RESEARCH INSTITUTE (US) 2008-08-12 US disclosed
US-5840991-A 3,4,5-TRIHYDROXYBENZYL-4-HYDROXYPHENYL THIOETHER DEVELOPMENT CENTER FOR BIOTECHNOLOGY (TW) 1998-11-24 US disclosed