SCHEMBL8536624

SCHEMBL8536624

CC(=O)C(CC(=O)c1ccc(C(C)(C)C)cc1)C(=O)O

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.55
MAPT P10636 3/20 0.55
NPSR1 Q6W5P4 2/20 0.55
LMNA P02545 4/20 0.53
HSP90AA1 P07900 1/20 0.53
THRB P10828 1/20 0.53
RAB9A P51151 4/20 0.51
NPC1 O15118 3/20 0.51
APAF1 O14727 1/20 0.48
RECQL P46063 2/20 0.48
HSD17B10 Q99714 2/20 0.47
ALOX15 P16050 1/20 0.47
APEX1 P27695 1/20 0.47
MAPK1 P28482 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
SRD5A2 P31213 1/20 0.47
HDAC1 Q13547 1/20 0.44
RARB P10826 1/20 0.44
RARG P13631 1/20 0.44
KDM4E B2RXH2 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8535820 0.83 ALDH1A1 (0.46) ALDH1A1MAPTNPSR1LMNAHSP90AA1
SCHEMBL11204474 0.81 ALDH1A1 (0.56) ALDH1A1MAPTNPSR1LMNAHSP90AA1
SCHEMBL10645702 0.80 TSHR (0.62) ALDH1A1MAPTNPSR1LMNARAB9A
SCHEMBL11014128 0.79 MAPT (0.58) ALDH1A1MAPTNPSR1LMNAHSP90AA1
SCHEMBL919272 0.74 GSK3B (0.66) ALDH1A1MAPTLMNARAB9ANPC1
SCHEMBL3823835 0.74 RAB9A (0.52) ALDH1A1MAPTNPSR1LMNAHSP90AA1
SCHEMBL7079689 0.74 RAB9A (0.66) ALDH1A1MAPTLMNARAB9ANPC1
SCHEMBL450084 0.74 RAB9A (0.85) ALDH1A1MAPTLMNARAB9ANPC1
SCHEMBL19642328 0.74 PDPK1 (0.65) ALDH1A1MAPTSRD5A2HDAC1TSHR
SCHEMBL14739209 0.73 ALDH1A1 (0.55) ALDH1A1MAPTNPSR1LMNAHSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0885869-A1 THERAPEUTIC AGENT FOR DIABETES Japan Tobacco Inc. (JP) 1998-12-23 EP disclosed