SCHEMBL8538568

SCHEMBL8538568

N=C(N)Nc1cccc(/C(CCc2ccccc2)=C(\CNC=O)C(=O)O)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.46
HPGD P15428 1/20 0.46
MAPT P10636 5/20 0.45
GAA P10253 3/20 0.45
RAB9A P51151 2/20 0.44
NPC1 O15118 1/20 0.44
ITGB3 P05106 1/20 0.42
ITGA2B P08514 1/20 0.42
HTT P42858 1/20 0.40
SENP1 Q9P0U3 1/20 0.39
ALOX15 P16050 1/20 0.39
SIRT2 Q8IXJ6 1/20 0.38
SIRT1 Q96EB6 1/20 0.38
SIRT3 Q9NTG7 1/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
LMNA P02545 1/20 0.38
ALOX12 P18054 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8541231 0.84 PARP1 (0.40) ALDH1A1HPGDRAB9ANPC1MEN1
SCHEMBL8542589 0.74 KMT2A (0.43) ALDH1A1RAB9ANPC1ITGB3ITGA2B
SCHEMBL7861970 0.70 ITGB3 (0.76) ALDH1A1ITGB3ITGA2BSIRT1KMT2A
SCHEMBL7373419 0.69 ITGB3 (0.66) ALDH1A1NPC1ITGB3ITGA2BMEN1
SCHEMBL7375114 0.69 ITGB3 (0.51) ALDH1A1HPGDITGB3ITGA2B
SCHEMBL8544650 0.69 PARP1 (0.42) ALDH1A1RAB9ASIRT1MEN1KMT2A
SCHEMBL7496410 0.68 PKM (0.53) ALDH1A1MAPTITGB3ITGA2BSIRT1
SCHEMBL7496407 0.68 PKM (0.53) ALDH1A1MAPTITGB3ITGA2BSIRT1
SCHEMBL5354517 0.68 L3MBTL1 (0.60) ALDH1A1MAPTGAARAB9AHTT
SCHEMBL7450519 0.68 PPARG (0.65) ALDH1A1HPGDRAB9ANPC1ITGB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5852210-A Cinnamic acid derivatives G. D. SEARLE & CO. (US) 1998-12-22 US claimed
US-5852210-A Cinnamic acid derivatives G. D. SEARLE & CO. (US) 1998-12-22 US disclosed