SCHEMBL8540341

SCHEMBL8540341

Fc1ccc2c(c1)C(c1ccccc1)CN2

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 1/20 0.42
SLC6A4 P31645 1/20 0.42
SLC6A3 Q01959 1/20 0.42
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
CYP3A4 P08684 2/20 0.40
CYP2D6 P10635 1/20 0.40
CYP19A1 P11511 1/20 0.39
DRD1 P21728 5/20 0.39
TACR2 P21452 1/20 0.38
CHRNB2 P17787 1/20 0.38
CHRNB4 P30926 1/20 0.38
CHRNA3 P32297 1/20 0.38
CHRNA4 P43681 1/20 0.38
TAAR1 Q96RJ0 1/20 0.37
KDM4E B2RXH2 3/20 0.37
DRD5 P21918 2/20 0.37
MAPT P10636 2/20 0.37
DRD2 P14416 2/20 0.37
HPGD P15428 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31694098 0.80 SIRT2 (0.44) MEN1KMT2ACYP3A4CYP2D6CYP19A1
SCHEMBL8537530 0.80 DRD1 (0.56) MEN1KMT2ACYP3A4CYP2D6DRD1
SCHEMBL20850872 0.80 DRD1 (0.43) MEN1KMT2ACYP3A4CYP2D6DRD1
SCHEMBL8543734 0.80 HTR2A (0.46) SLC6A2SLC6A4SLC6A3MEN1KMT2A
SCHEMBL11547755 0.80 ALOX12 (0.43) SLC6A3MEN1KMT2ACYP3A4CYP2D6
SCHEMBL5871368 0.79 PRCP (0.42) MEN1KMT2ACYP3A4CYP2D6MAPT
SCHEMBL4001774 0.78 MEN1 (0.52) MEN1KMT2ACYP3A4CYP2D6DRD1
SCHEMBL2347871 0.78 SLC6A2 (0.46) SLC6A2SLC6A4SLC6A3MEN1KMT2A
SCHEMBL8482343 0.77 PKM (0.43) SLC6A2SLC6A4SLC6A3KDM4EMAPT
Hydrochloric Acid SCHEMBL11553849 0.77 MEN1 (0.50) MEN1KMT2ACYP3A4CYP2D6DRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0721949-B1 INDOLINE COMPOUND AND 5-HT 3? RECEPTOR ANTAGONIST CONTAINING THE SAME AS ACTIVE INGREDIENT TOKYO TANABE CO (JP) 1998-01-07 EP disclosed
US-5677326-A GASTROINTESTINAL DISORDERS TOKYO TANABE COMPANY LIMITED (JP) 1997-10-14 US disclosed
EP-0721949-A1 INDOLINE COMPOUND AND 5-HT 3? RECEPTOR ANTAGONIST CONTAINING THE SAME AS ACTIVE INGREDIENT TOKYO TANABE COMPANY LIMITED (JP) 1996-07-17 EP disclosed