SCHEMBL8545748

SCHEMBL8545748

CCN(CC)S(=O)(=O)c1ccc(OC)c(-c2ccc[nH]2)c1

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.54
MAPT P10636 1/20 0.54
KDM4E B2RXH2 2/20 0.50
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
DRD2 P14416 1/20 0.46
DRD3 P35462 1/20 0.46
RXFP1 Q9HBX9 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
KMT2A Q03164 3/20 0.45
LMNA P02545 2/20 0.45
MEN1 O00255 2/20 0.45
RECQL P46063 1/20 0.44
POLB P06746 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8540116 0.90 L3MBTL1 (0.55) ALDH1A1MAPTKDM4EDRD2DRD3
SCHEMBL9052649 0.90 DRD2 (0.54) ALDH1A1KDM4EDRD2DRD3SMN1; SMN2
SCHEMBL9053369 0.89 DRD2 (0.52) ALDH1A1MAPTKDM4EDRD2DRD3
SCHEMBL8544314 0.86 MAPT (0.54) ALDH1A1MAPTKDM4EDRD2DRD3
SCHEMBL9053438 0.85 SMN1; SMN2 (0.51) ALDH1A1MAPTKDM4EDRD2DRD3
SCHEMBL8544972 0.84 DRD2 (0.56) DRD2DRD3
SCHEMBL9053373 0.81 DRD2 (0.50) ALDH1A1MAPTKDM4EDRD2DRD3
SCHEMBL9053622 0.81 DRD2 (0.50) MAPTKDM4EDRD2DRD3SMN1; SMN2
SCHEMBL9053039 0.79 PGR (0.51) ALDH1A1MAPTKDM4ECYP1A2CYP3A4
SCHEMBL8540314 0.78 POLB (0.47) ALDH1A1MAPTKDM4EDRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0705259-B1 PHENYRROLE DERIVATIVES AND THEIR USE AS DOPAMINE D3 ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1998-02-25 EP disclosed
EP-0705259-A1 PHENYRROLE DERIVATIVES AND THEIR USE AS DOPAMINE D3 ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1996-04-10 EP disclosed
WO-1995000508-A1 PHENYRROLE DERIVATIVES AND THEIR USE AS DOPAMINE D3 ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1995-01-05 WO disclosed