SCHEMBL8549480

SCHEMBL8549480

NC(=S)CCC1CCN(OCc2ccccc2)C(=C=O)C1

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
BCHE P06276 2/20 0.35
ACHE P22303 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
CYP2C19 P33261 1/20 0.35
NPC1 O15118 1/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
MGLL Q99685 1/20 0.33
GRIN2B Q13224 2/20 0.33
CTSL P07711 1/20 0.33
CTSB P07858 1/20 0.33
CTSK P43235 1/20 0.33
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
LMNA P02545 1/20 0.32
MAPT P10636 1/20 0.32
MAPK1 P28482 1/20 0.32
TDP1 Q9NUW8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7747533 0.78 ITGB3 (0.46) SMN1; SMN2CYP2C19NPC1CYP2D6CYP2C9
SCHEMBL7398369 0.77 GRIN2B (0.35) MEN1KMT2AGRIN2BCYP2D6CYP2C9
SCHEMBL7448545 0.76 SMN1; SMN2 (0.53) SMN1; SMN2CYP2C19NPC1MEN1KMT2A
SCHEMBL7403343 0.75 CTSL (0.36) CTSLCTSBCTSK
SCHEMBL9796122 0.72 ALDH1A1 (0.38) BCHESMN1; SMN2CYP2C19NPC1
SCHEMBL8552418 0.72 MGLL (0.35) BCHEACHESMN1; SMN2CYP2C19NPC1
SCHEMBL8549475 0.71 SMN1; SMN2 (0.65) SMN1; SMN2CYP2C19NPC1MEN1KMT2A
SCHEMBL8552420 0.71 BCHE (0.45) BCHEACHELMNA
SCHEMBL9204131 0.70 CTSL (0.36) MEN1KMT2ACTSLCTSBCTSK
SCHEMBL27613312 0.70 KDM4E (0.36) SMN1; SMN2KMT2AGRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0858457-A1 5-MEMBERED HETEROCYCLES, PHARMACEUTICAL AGENTS CONTAINING SAID COMPOUNDS AND THE USE THEREOF AND METHODS OF PRODUCING THEM Dr. Karl Thomae GmbH (DE) 1998-08-19 EP disclosed
WO-1997015567-A1 5-MEMBERED HETEROCYCLES, PHARMACEUTICAL AGENTS CONTAINING SAID COMPOUNDS AND THE USE THEREOF AND METHODS OF PRODUCING THEM DR. KARL THOMAE GMBH (DE) 1997-05-01 WO disclosed