SCHEMBL8549583

SCHEMBL8549583

CCCCN(CCCC)S(=O)(=O)Nc1ccc2oc(C)c(CCN(C)Cc3ncc([N+](=O)[O-])cn3)c2c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HIF1A Q16665 2/20 0.39
ESR1 P03372 1/20 0.34
PGR P06401 1/20 0.34
CHRM2 P08172 1/20 0.34
HTR1A P08908 1/20 0.34
ADRA2A P08913 1/20 0.34
ADORA3 P0DMS8 1/20 0.34
CHRM1 P11229 1/20 0.34
DRD1 P21728 1/20 0.34
TBXA2R P21731 1/20 0.34
SLC6A2 P23975 1/20 0.34
PDE4A P27815 1/20 0.34
SLC6A4 P31645 1/20 0.34
ADRA1A P35348 1/20 0.34
OPRM1 P35372 1/20 0.34
DRD3 P35462 1/20 0.34
SLC6A3 Q01959 1/20 0.34
KCNH2 Q12809 1/20 0.34
HRH3 Q9Y5N1 1/20 0.34
LMNA P02545 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7146368 0.84 ALDH1A1 (0.38) HTR1AADRA2ASLC6A2KCNH2LMNA
SCHEMBL8694248 0.84 MAPT (0.33) HIF1ALMNAMAPTHTTMEN1
SCHEMBL8548197 0.70 HTT (0.32) HTT
SCHEMBL8547960 0.69 ALDH1A1 (0.31)
Acetic Acid SCHEMBL8552677 0.68 MEN1 (0.36) MAPTTP53MEN1KMT2A
SCHEMBL8548340 0.65 HTT (0.43) LMNAMAPTHTTPOLBMEN1
SCHEMBL8553359 0.65 HIF1A (0.42) HIF1ALMNAMAPTHTTMEN1
SCHEMBL5329933 0.63 HTT (0.45) LMNAMAPTHTTMEN1KMT2A
SCHEMBL8550195 0.63 MEN1 (0.44) HIF1AMAPTTP53POLBMEN1
SCHEMBL8552248 0.62 CNR1 (0.47) MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5792763-A MIGRAINES; ANALGESICS; DISEASES LINKED TO DECREASED NEUROTRANMISSION OF SEROTONIN IN MAMMALS ELI LILLY AND COMPANY (US) 1998-08-11 US disclosed
EP-0835869-A2 New serotonin 5-HT1F agonists ELI LILLY AND COMPANY (US) 1998-04-15 EP disclosed