SCHEMBL8549838

SCHEMBL8549838

CC(=O)Nc1ccc2oc(C)c(CCN(C)C)c2c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.47
HPGD P15428 5/20 0.47
KDM4E B2RXH2 4/20 0.47
HSD17B10 Q99714 3/20 0.47
MAPT P10636 3/20 0.47
ALOX15 P16050 2/20 0.47
TSHR P16473 2/20 0.47
PKM P14618 1/20 0.47
MAPK1 P28482 1/20 0.47
HTR1F P30939 2/20 0.44
CA12 O43570 2/20 0.43
CA9 Q16790 2/20 0.43
CA1 P00915 1/20 0.43
HRH3 Q9Y5N1 1/20 0.40
NPC1 O15118 1/20 0.39
TP53 P04637 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
CSNK2A2 P19784 1/20 0.39
CSNK2B P67870 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8692074 0.85 HPGD (0.45) ALDH1A1HPGDKDM4EMAPTMAPK1
SCHEMBL8551309 0.85 RAB9A (0.48) ALDH1A1KDM4EHTR1FNPC1RAB9A
SCHEMBL8549636 0.83 HTR1F (0.51) ALDH1A1HPGDKDM4EHSD17B10MAPT
SCHEMBL8547488 0.83 HTR1F (0.53) HSD17B10MAPTHTR1FCA12CA9
SCHEMBL8552580 0.83 HTR1F (0.65) ALDH1A1KDM4EMAPTHTR1FNPC1
SCHEMBL8548295 0.82 RAB9A (0.51) ALDH1A1HPGDKDM4EHSD17B10MAPT
SCHEMBL8552436 0.81 KMT2A (0.49) ALDH1A1HPGDKDM4EHSD17B10MAPT
SCHEMBL8552089 0.81 HTR1F (0.52) MAPTHTR1FNPC1TP53RAB9A
SCHEMBL8549211 0.81 HTR1F (0.49) ALDH1A1KDM4EMAPTMAPK1HTR1F
SCHEMBL8709033 0.79 HTR1F (0.48) MAPTHTR1FNPC1TP53RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5792763-A MIGRAINES; ANALGESICS; DISEASES LINKED TO DECREASED NEUROTRANMISSION OF SEROTONIN IN MAMMALS ELI LILLY AND COMPANY (US) 1998-08-11 US disclosed
EP-0835869-A2 New serotonin 5-HT1F agonists ELI LILLY AND COMPANY (US) 1998-04-15 EP disclosed