SCHEMBL8550889

SCHEMBL8550889

Cc1sc2ccc(NS(=O)(=O)c3ccccc3)cc2c1CCN(C)Cc1ccc2ccncc2c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 4/20 0.38
ROCK1 Q13464 3/20 0.38
IKBKB O14920 2/20 0.38
JAK2 O60674 2/20 0.38
ROCK2 O75116 2/20 0.38
JAK3 P52333 2/20 0.38
LMNA P02545 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
ALDH1A1 P00352 3/20 0.36
HPGD P15428 1/20 0.36
ADRB2 P07550 2/20 0.35
ADRB1 P08588 2/20 0.35
ADRB3 P13945 2/20 0.35
IMPDH2 P12268 1/20 0.35
NAMPT P43490 1/20 0.35
CYP17A1 P05093 1/20 0.35
ITK Q08881 1/20 0.34
PDE4A P27815 1/20 0.34
PDE4B Q07343 1/20 0.34
PDE4C Q08493 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7138773 0.84 IMPDH2 (0.45) HTR6ROCK1IKBKBJAK2ROCK2
SCHEMBL8550195 0.84 MEN1 (0.44) HTR6ROCK1IKBKBJAK2ROCK2
SCHEMBL8547927 0.75 ROCK1 (0.37) ROCK1ROCK2LMNASMN1; SMN2ALDH1A1
SCHEMBL8549554 0.73 HTR6 (0.42) HTR6LMNASMN1; SMN2ALDH1A1
SCHEMBL12922863 0.67 BRD4 (0.50) HTR6LMNASMN1; SMN2ALDH1A1HPGD
SCHEMBL10356533 0.67 LMNA (0.69) ROCK1IKBKBJAK2ROCK2JAK3
SCHEMBL8554008 0.65 BRAF (0.30)
SCHEMBL8191020 0.62 HTR1F (0.42) LMNASMN1; SMN2ALDH1A1ITK
SCHEMBL8552127 0.62 KDM4E (0.39) ROCK1ROCK2LMNASMN1; SMN2ALDH1A1
SCHEMBL17437173 0.62 LMNA (0.56) HTR6ROCK1IKBKBJAK2ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998015545-A1 NEW SEROTONIN 5-HT1F AGONISTS ELI LILLY AND COMPANY (US) 1998-04-16 WO disclosed
EP-0835869-A2 New serotonin 5-HT1F agonists ELI LILLY AND COMPANY (US) 1998-04-15 EP disclosed