SCHEMBL8552270

SCHEMBL8552270

O=C(Cc1cccc(Cl)c1Cl)N(O)C[C@@H](c1ccccc1)N1CC[C@H](O)C1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 4/20 0.43
SLC6A4 P31645 4/20 0.43
CCR5 P51681 2/20 0.43
CACNA2D1 P54289 1/20 0.39
CACNA1B Q00975 1/20 0.39
CACNB1 Q02641 1/20 0.39
CACNA1C Q13936 1/20 0.39
HTR1D P28221 2/20 0.38
HTR1B P28222 2/20 0.38
OPRK1 P41145 4/20 0.37
CYP2D6 P10635 2/20 0.37
SLC6A3 Q01959 2/20 0.37
CYP3A4 P08684 1/20 0.37
KCNH2 Q12809 1/20 0.37
TACR1 P25103 1/20 0.37
OPRM1 P35372 1/20 0.36
OPRD1 P41143 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8551509 0.90 SIGMAR1 (0.39) SLC6A2SLC6A4CCR5CACNA2D1CACNA1B
SCHEMBL8547882 0.86 CCR5 (0.43) SLC6A2SLC6A4CCR5CACNA2D1CACNA1B
SCHEMBL8553707 0.84 CCR5 (0.48) CCR5CACNA2D1CACNA1BCACNB1CACNA1C
SCHEMBL8550877 0.83 CCR5 (0.51) CCR5OPRK1CYP2D6CYP3A4OPRM1
SCHEMBL8552457 0.80 CCR5 (0.48) CCR5OPRK1CYP2D6TACR1OPRM1
SCHEMBL8551862 0.77 TACR1 (0.41) CCR5OPRK1CYP2D6TACR1OPRM1
SCHEMBL6973106 0.76 OPRK1 (0.53) CCR5OPRK1CYP2D6OPRM1OPRD1
SCHEMBL6973107 0.76 OPRK1 (0.53) CCR5OPRK1CYP2D6OPRM1OPRD1
SCHEMBL8476568 0.74 CCR5 (0.43) CCR5OPRK1CYP2D6CYP3A4TACR1
SCHEMBL8552339 0.73 NOTUM (0.44) CCR5KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0817772-A1 PYRROLIDINYL HYDROXAMIC ACID COMPOUNDS AND THEIR PRODUCTION PROCESS PFIZER INC. (US) 1998-01-14 EP claimed
EP-0817772-A1 PYRROLIDINYL HYDROXAMIC ACID COMPOUNDS AND THEIR PRODUCTION PROCESS PFIZER INC. (US) 1998-01-14 EP disclosed