SCHEMBL8553051

SCHEMBL8553051

O=C(F)c1ccc(N2CCNCC2)c(F)c1F

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 8/20 0.45
DRD2 P14416 2/20 0.39
DRD3 P35462 2/20 0.39
DRD1 P21728 1/20 0.39
HTR2A P28223 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
HTR7 P34969 1/20 0.39
ADRB1 P08588 2/20 0.39
DRD4 P21917 1/20 0.38
ALDH1A1 P00352 2/20 0.38
LMNA P02545 1/20 0.38
KDR P35968 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25366356 0.86 HTR6 (0.44) HTR6DRD2DRD3DRD1HTR2A
SCHEMBL25232509 0.79 ALDH1A1 (0.45) HTR6ADRB1ALDH1A1LMNA
SCHEMBL20076208 0.78 HTR6 (0.46) HTR6HTR7ALDH1A1LMNAKDR
SCHEMBL8191985 0.75 HTR1A (0.46) HTR6DRD2DRD3HTR2ASIGMAR1
Hydrochloric Acid SCHEMBL15937978 0.74 LMNA (0.48) HTR6SIGMAR1HTR7ADRB1ALDH1A1
SCHEMBL4420344 0.73 HTR6 (0.46) HTR6HTR7ADRB1
SCHEMBL26968308 0.73 TTR (0.57) HTR6DRD2DRD3HTR2ASIGMAR1
SCHEMBL29835980 0.73 TTR (0.57) HTR6DRD2DRD3HTR2ASIGMAR1
SCHEMBL31342302 0.73 HTR6 (0.57) HTR6HTR2AHTR7ADRB1ALDH1A1
SCHEMBL24632769 0.73 ADRB1 (0.55) HTR7ADRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0836599-A1 1,6-DISUBSTITUTED ISOCHROMANS FOR TREATMENT OF MIGRAINE HEADACHES PHARMACIA & UPJOHN COMPANY (US) 1998-04-22 EP disclosed
WO-1997002259-A1 1,6-DISUBSTITUTED ISOCHROMANS FOR TREATMENT OF MIGRAINE HEADACHES PHARMACIA & UPJOHN COMPANY (US) 1997-01-23 WO disclosed